Compile Data Set for Download or QSAR
Found 308 with Last Name = 'duroux' and Initial = 'r'
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50144221(CHEMBL3759802)copy SMILEScopy InChI
Affinity DataKi:  0.0900nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464407(CHEMBL4292336)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464406(CHEMBL4280601)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464415(CHEMBL4278575)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464420(CHEMBL4290302)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50037242(CHEMBL323332 | N-(2-(5-methoxybenzofuran-3-yl)ethy...)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464400(CHEMBL4293386)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464409(CHEMBL4283539)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464414(CHEMBL4288497)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464413(CHEMBL4281712)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464403(CHEMBL4294790)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464417(CHEMBL4280791)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464411(CHEMBL4291381)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.210nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.230nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464421(CHEMBL4286896)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464415(CHEMBL4278575)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464400(CHEMBL4293386)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464418(CHEMBL4284223)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50037242(CHEMBL323332 | N-(2-(5-methoxybenzofuran-3-yl)ethy...)copy SMILEScopy InChI
Affinity DataKi:  0.340nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464399(CHEMBL4278446)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464404(CHEMBL4286494)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464408(CHEMBL4285145)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464416(CHEMBL4289115)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464413(CHEMBL4281712)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50144222(CHEMBL3758717)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))TBA
LigandPNGBDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44V8SPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))TBA
LigandPNGBDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5XPZPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.520nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50144226(CHEMBL3758679)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464407(CHEMBL4292336)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464414(CHEMBL4288497)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50144310(CHEMBL3759084)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50144219(CHEMBL3758225)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464421(CHEMBL4286896)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50464419(CHEMBL4277185)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464406(CHEMBL4280601)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50144368(CHEMBL3759372)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464409(CHEMBL4283539)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
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