TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of RANTES-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Antagonist activity at CCR1 receptor in human THP1 cells assessed as inhibition of MIP-1alpha induced chemotaxis after 60 minsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MPIF-1-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 2.90nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Bristol-Myers Squibb Company
Affinity DataIC50: 3nMAssay Description:The enzyme was assayed with substrate GST-Rb in the presence of 50 uM ATP/[gamma-32P] ATP, and capturing the 32-P labeled reaction products on GSH-Se...More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MIP-1alpha from CCR1 in human THP1 cellsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at CCR1 receptor in human THP1 cells assessed as inhibition of MIP-1alpha induced chemotaxis after 60 minsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at CCR1 receptor in human THP1 cells assessed as inhibition of HCC4-induced chemotaxis after 60 minsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Antagonist activity at CCR1 receptor in human THP1 cells assessed as inhibition of RANTES-induced chemotaxis after 60 minsMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Bristol-Myers Squibb Company
Curated by ChEMBL
Bristol-Myers Squibb Company
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
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