Affinity DataKi: 0.0126nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0158nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0251nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0398nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
Affinity DataKi: 0.0501nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.0631nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0631nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibitory affinity constant (pKi) against tachykinin receptor 2 (NK-2R) using heterologous competition experimentsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of 125I-cyanopindolol from human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Binding affinity towards Tachykinin receptor 2More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]-N-methylscopolamine from human muscarinic M3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-N-methylscopolamine from human muscarinic M3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:In vitro functional activity towards Neurokinin NK2 receptor on isolated rabbit urinary bladder (RUB)More data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.126nMAssay Description:Displacement of [125I]neurokinin A from human NK2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-N-methylscopolamine from human muscarinic M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-N-methylscopolamine from human muscarinic M3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.158nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M2 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Maryland
Curated by ChEMBL
University of Maryland
Curated by ChEMBL