Compile Data Set for Download or QSAR
Found 34 with Last Name = 'ruzziconi' and Initial = 'r'
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153269(CHEMBL3775575)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153186(CHEMBL3774520)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153316(CHEMBL3775207)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153183(CHEMBL3774548)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153314(CHEMBL3774689)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153284(CHEMBL3775852)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153278(CHEMBL3775105)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153317(CHEMBL3774886)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153187(CHEMBL3775401)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153271(CHEMBL3774968)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153268(CHEMBL3775173)copy SMILEScopy InChI
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153270(CHEMBL3775819)copy SMILEScopy InChI
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153272(CHEMBL3775722)copy SMILEScopy InChI
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153283(CHEMBL3774445)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153182(CHEMBL3775053)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153285(CHEMBL3774995)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153185(CHEMBL3775726)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153184(CHEMBL3774891)copy SMILEScopy InChI
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153192(CHEMBL3775789)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153277(CHEMBL3774527)copy SMILEScopy InChI
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153288(CHEMBL3775693)copy SMILEScopy InChI
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153279(CHEMBL3775483)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153274(CHEMBL3775322)copy SMILEScopy InChI
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153280(CHEMBL3774675)copy SMILEScopy InChI
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153281(CHEMBL3775062)copy SMILEScopy InChI
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153282(CHEMBL3775841)copy SMILEScopy InChI
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153315(CHEMBL3774582)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153249(CHEMBL3775871)copy SMILEScopy InChI
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153247(CHEMBL3775857)copy SMILEScopy InChI
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153276(CHEMBL3775445)copy SMILEScopy InChI
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153275(CHEMBL3775842)copy SMILEScopy InChI
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153286(CHEMBL3775271)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153287(CHEMBL3775507)copy SMILEScopy InChI
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
University of Perugia

Curated by ChEMBL
LigandPNGBDBM50153273(CHEMBL3775114)copy SMILEScopy InChI
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of NorA efflux pump in Staphylococcus aureus 1199B assessed as reduction in EtBr efflux incubated for 20 mins measured for 5 mins by real-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28W3G57PubMed