Compile Data Set for Download or QSAR
Found 372 with Last Name = 'sasaki' and Initial = 'r'
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444909(CHEMBL3099618)copy SMILEScopy InChI
Affinity DataKi:  340nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444909(CHEMBL3099618)copy SMILEScopy InChI
Affinity DataKi:  580nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444908(CHEMBL3099624)copy SMILEScopy InChI
Affinity DataKi:  670nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444908(CHEMBL3099624)copy SMILEScopy InChI
Affinity DataKi:  870nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444888(CHEMBL3099621)copy SMILEScopy InChI
Affinity DataKi:  1.02E+3nMAssay Description:Competitive inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate Linewea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444888(CHEMBL3099621)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Noncompetitive inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogeni...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of PGPH activity of human 26S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50432548(LACTACYSTIN)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50324535(3-{[9-(Dimethylamino)nonanoyl](hydroxy)amino}propa...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of KDM2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458013(CHEMBL4215864)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444899(CHEMBL3099640)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458009(CHEMBL4205518)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444904(CHEMBL3099622)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50121213(CHEMBL3622371)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human LSD1 using H3K4 peptide as substrate by peroxidase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TWVPubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444909(CHEMBL3099618)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444889(CHEMBL3099620)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458008(CHEMBL4204198)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444907(CHEMBL3099623)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458009(CHEMBL4205518)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444908(CHEMBL3099624)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444888(CHEMBL3099621)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50140044(CHEMBL3764353)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of human LSD1 using H3K4 peptide as substrate by peroxidase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TWVPubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444909(CHEMBL3099618)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50140043(CHEMBL3765529)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of human LSD1 using H3K4 peptide as substrate by peroxidase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TWVPubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444908(CHEMBL3099624)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50140045(CHEMBL3764836)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Inhibition of human LSD1 using H3K4 peptide as substrate by peroxidase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TWVPubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444906(CHEMBL3099636)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444909(CHEMBL3099618)copy SMILEScopy InChI
Affinity DataIC50: 640nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444906(CHEMBL3099636)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444908(CHEMBL3099624)copy SMILEScopy InChI
Affinity DataIC50: 690nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50069989((R)-3-methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxa...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444909(CHEMBL3099618)copy SMILEScopy InChI
Affinity DataIC50: 720nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444901(CHEMBL3099638)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444901(CHEMBL3099638)copy SMILEScopy InChI
Affinity DataIC50: 770nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444885(CHEMBL3099637)copy SMILEScopy InChI
Affinity DataIC50: 790nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50324535(3-{[9-(Dimethylamino)nonanoyl](hydroxy)amino}propa...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of KDM4A (unknown origin) using H3K9me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB475VPubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444885(CHEMBL3099637)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444903(CHEMBL3099631)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444907(CHEMBL3099623)copy SMILEScopy InChI
Affinity DataIC50: 870nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444905(CHEMBL3099635)copy SMILEScopy InChI
Affinity DataIC50: 880nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome beta 2 subunit assessed as hydrolysis of Boc-LRR-AMC fluorogenic substrate measured for 1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458007(CHEMBL4209883)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458014(CHEMBL4206039)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444898(CHEMBL3099625)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458004(CHEMBL4210397)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50458014(CHEMBL4206039)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TV7PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444907(CHEMBL3099623)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as hydrolysis of succinyl-LLVY-AMC fluorogenic substrate mea...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Institute of Bio-Science and Technology

Curated by ChEMBL
LigandPNGBDBM50444905(CHEMBL3099635)copy SMILEScopy InChI
Affinity DataIC50: 910nMAssay Description:Inhibition of PGPH-like activity of human 20S proteasome beta 1 subunit assessed as hydrolysis of Z-LLE-AMC fluorogenic substrate measured for 1 hr b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222W81PubMed
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