Compile Data Set for Download or QSAR
Found 294 with Last Name = 'sawa' and Initial = 'r'
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Institute for Theoretical Medicine, Inc.

Curated by ChEMBL
LigandPNGBDBM50330795(2-hydroxy-5-isopropyl-2,4,6-cycloheptatrien-1-one ...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Competitive inhibition of mushroom tyrosinase after 15 mins by Lineweaver-Bulk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3MF5PubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Institute for Theoretical Medicine, Inc.

Curated by ChEMBL
LigandPNGBDBM50330794(2-Hydroxy-4-isopropyl-cyclohepta-2,4,6-trienone | ...)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Competitive inhibition of mushroom tyrosinase after 15 mins by Lineweaver-Bulk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3MF5PubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Institute for Theoretical Medicine, Inc.

Curated by ChEMBL
LigandPNGBDBM50330793(2-hydroxy-3-isopropyl-2,4,6-cycloheptatrien-1-one ...)copy SMILEScopy InChI
Affinity DataKi:  3.30E+3nMAssay Description:Competitive inhibition of mushroom tyrosinase after 15 mins by Lineweaver-Bulk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3MF5PubMed
TargetNeprilysin(Homo sapiens (Human))
Kao Corporation

Curated by ChEMBL
LigandPNGBDBM50354041(CHEMBL1829584)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:Inhibition of neutral endopeptidase in human fibroblasts homogenates using glutaryl-Ala-Ala-Phe-4-methoxy-2-naphtylamide as substrate after 1 hrs by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154HF6PubMed
TargetNeprilysin(Homo sapiens (Human))
Kao Corporation

Curated by ChEMBL
LigandPNGBDBM50354042(CHEMBL1829585)copy SMILEScopy InChI
Affinity DataIC50: 0.510nMAssay Description:Inhibition of neutral endopeptidase in human fibroblasts homogenates using glutaryl-Ala-Ala-Phe-4-methoxy-2-naphtylamide as substrate after 1 hrs by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154HF6PubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of Flt4 (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetNeprilysin(Homo sapiens (Human))
Kao Corporation

Curated by ChEMBL
LigandPNGBDBM50251742((3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyl-tetrahydro...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of neutral endopeptidase in human fibroblasts homogenates using glutaryl-Ala-Ala-Phe-4-methoxy-2-naphtylamide as substrate after 1 hrs by ...More data for this Ligand-Target Pair
TargetNeprilysin(Homo sapiens (Human))
Kao Corporation

Curated by ChEMBL
LigandPNGBDBM50354040(CHEMBL1829583)copy SMILEScopy InChI
Affinity DataIC50: 9.70nMAssay Description:Inhibition of neutral endopeptidase in human fibroblasts homogenates using glutaryl-Ala-Ala-Phe-4-methoxy-2-naphtylamide as substrate after 1 hrs by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154HF6PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50362881(CHEMBL1940907)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant GSK3-beta after 1 hr by KinaseGlo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0FXVPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of KDR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of GST-Flt1 kinase domain (unknown origin) expressed in baculovirus infected Sf9 cells after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50325983(6-(2-(4-(2,4-dichlorophenyl)-5-(4-methyl-1H-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50325983(6-(2-(4-(2,4-dichlorophenyl)-5-(4-methyl-1H-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant GSK3-beta after 1 hr by KinaseGlo luciferase assayMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50362879(CHEMBL1940905)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of human recombinant GSK3-beta after 1 hr by KinaseGlo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0FXVPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50362880(CHEMBL1940906)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant GSK3-beta after 1 hr by KinaseGlo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0FXVPubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Institute for Theoretical Medicine, Inc.

Curated by ChEMBL
LigandPNGBDBM50330795(2-hydroxy-5-isopropyl-2,4,6-cycloheptatrien-1-one ...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of mushroom tyrosinase after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3MF5PubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Institute for Theoretical Medicine, Inc.

Curated by ChEMBL
LigandPNGBDBM50330794(2-Hydroxy-4-isopropyl-cyclohepta-2,4,6-trienone | ...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of mushroom tyrosinase after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3MF5PubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of PDGFR-alpha (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50362882(CHEMBL1940908)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant GSK3-beta after 1 hr by KinaseGlo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0FXVPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50362878(CHEMBL1940904)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant GSK3-beta after 1 hr by KinaseGlo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0FXVPubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of PDGFR-beta (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetNeprilysin(Homo sapiens (Human))
Kao Corporation

Curated by ChEMBL
LigandPNGBDBM50354044(CHEMBL1829587)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of neutral endopeptidase in human fibroblasts homogenates using glutaryl-Ala-Ala-Phe-4-methoxy-2-naphtylamide as substrate after 1 hrs by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154HF6PubMed
TargetNeprilysin(Homo sapiens (Human))
Kao Corporation

Curated by ChEMBL
LigandPNGBDBM50354043(CHEMBL1829586)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of neutral endopeptidase in human fibroblasts homogenates using glutaryl-Ala-Ala-Phe-4-methoxy-2-naphtylamide as substrate after 1 hrs by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2154HF6PubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of PDGFR-beta (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of Flt4 (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50362883(CHEMBL1940909)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of human recombinant GSK3-beta after 1 hr by KinaseGlo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0FXVPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM15236(3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chr...)copy SMILEScopy InChI
Affinity DataIC50: 560nMAssay Description:Inhibition of human recombinant His-tagged Glyoxalase 1 expressed in Sf21-Baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z037XFPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM15236(3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chr...)copy SMILEScopy InChI
Affinity DataIC50: 560nMAssay Description:Inhibition of recombinant human His-tagged glyoxalase 1 expressed in Escherichia coli BL21 assessed as formation of S-D-lactoylglutathione after 5 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7J38PubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50045936((E)-4-(3,5-dihydroxystyryl)benzene-1,2-diol | (E)-...)copy SMILEScopy InChI
Affinity DataIC50: 760nMAssay Description:Inhibition of human N-terminal His6-tagged GLO1 expressed in baculovirus infected sf21 cells assessed as reduction in S-D-lactoylglutathione formatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0HQ0PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50326997(CHEMBL590878 | Delphinidin)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant glyoxalase 1 assessed as S-D-lactoylglutathione after 15 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC32K6PubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50355547(CHEMBL1910548)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human His-tagged glyoxalase 1 expressed in Escherichia coli BL21 assessed as formation of S-D-lactoylglutathione after 5 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7J38PubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569128(CHEMBL4853249)copy SMILES
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569120(CHEMBL4861582)copy SMILES
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of EGFR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569133(CHEMBL4875229)copy SMILES
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569134(CHEMBL4863408)copy SMILES
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of GST-Flt1 kinase domain (unknown origin) expressed in baculovirus infected Sf9 cells after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569131(CHEMBL4852940)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human recombinant His-tagged Glyoxalase 1 expressed in Sf21-Baculovirus systemMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z037XFPubMed
TargetDeoxyribonuclease gamma(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50206432(4-(4,6-dichloro-1,3,5-triazin-2-ylamino)-2-(6-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of human recombinant DNase gamma expressed in Rosetta DE3 cells assessed as increase in acidsoluble DNA after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0GDVPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569129(CHEMBL4851336)copy SMILES
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of PDGFR-alpha (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569125(CHEMBL4871220)copy SMILES
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569130(CHEMBL1303934)copy SMILES
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569127(CHEMBL4877301)copy SMILES
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569121(CHEMBL1162436)copy SMILES
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM54054((E)-3-(1,3-benzoxazol-2-yl)-4-(4-methoxyphenyl)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569132(CHEMBL4848220)copy SMILES
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University of Science

Curated by ChEMBL
LigandPNGBDBM50569124(CHEMBL4877073)copy SMILES
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of Glyoxalase-1 (unknown origin) assessed as inhibition of S-D-lactoylglutathione formation using MG and reduced glutathione as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0XNTPubMed
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