Compile Data Set for Download or QSAR
Found 550 with Last Name = 'sommer' and Initial = 'r'
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259915(US9512115, 19)copy SMILES
Affinity DataKi:  2.49nM ΔG°:  -49.9kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259915(US9512115, 19)copy SMILES
Affinity DataKi:  2.53nM ΔG°:  -49.9kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259914(US9512115, 18)copy SMILES
Affinity DataKi:  2.69nM ΔG°:  -49.7kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259898(US9512115, 1)copy SMILES
Affinity DataKi:  2.90nM ΔG°:  -49.5kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259914(US9512115, 18)copy SMILES
Affinity DataKi:  2.92nM ΔG°:  -49.5kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM149365(US8962860, 9)copy SMILES
Affinity DataKi:  3.24nM ΔG°:  -49.3kJ/mole IC50: 3.08nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856V2US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259907(US9512115, 11)copy SMILES
Affinity DataKi:  3.34nM ΔG°:  -49.2kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259898(US9512115, 1)copy SMILES
Affinity DataKi:  3.58nM ΔG°:  -49.0kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM149363(US8962860, 6)copy SMILES
Affinity DataKi:  3.80nM ΔG°:  -48.9kJ/mole IC50: 234nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856V2US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM149366(US8962860, 11)copy SMILES
Affinity DataKi:  4.13nM ΔG°:  -48.7kJ/mole IC50: 48nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856V2US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259916(US9512115, 20)copy SMILES
Affinity DataKi:  4.53nM ΔG°:  -48.4kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259900(US9512115, 3)copy SMILES
Affinity DataKi:  5.02nM ΔG°:  -48.2kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259900(US9512115, 3)copy SMILES
Affinity DataKi:  5.03nM ΔG°:  -48.2kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259919(US9512115, 23)copy SMILES
Affinity DataKi:  5.15nM ΔG°:  -48.1kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259916(US9512115, 20)copy SMILES
Affinity DataKi:  5.29nM ΔG°:  -48.0kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259907(US9512115, 11)copy SMILES
Affinity DataKi:  5.54nM ΔG°:  -47.9kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM50299853(1-(3,4-Dimethoxyphenyl)-3-(3-(5-methyl-1H-imidazol...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21Z46GVUS Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM149358(US8962860, 1)copy SMILES
Affinity DataKi:  6.07nM ΔG°:  -47.7kJ/mole IC50: 69.7nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856V2US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259903(US9512115, 6)copy SMILES
Affinity DataKi:  6.21nM ΔG°:  -47.6kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM149375(US8962860, 42)copy SMILES
Affinity DataKi:  6.49nM ΔG°:  -47.5kJ/mole IC50: 24nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856V2US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259899(US9512115, 2)copy SMILES
Affinity DataKi:  6.54nM ΔG°:  -47.5kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259913(US9512115, 17)copy SMILES
Affinity DataKi:  6.66nM ΔG°:  -47.4kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259903(US9512115, 6)copy SMILES
Affinity DataKi:  6.71nM ΔG°:  -47.4kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259919(US9512115, 23)copy SMILES
Affinity DataKi:  7.89nM ΔG°:  -47.0kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259913(US9512115, 17)copy SMILES
Affinity DataKi:  8.29nM ΔG°:  -46.9kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259899(US9512115, 2)copy SMILES
Affinity DataKi:  8.5nM ΔG°:  -46.8kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259906(US9512115, 10)copy SMILES
Affinity DataKi:  8.95nM ΔG°:  -46.7kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259906(US9512115, 10)copy SMILES
Affinity DataKi:  8.99nM ΔG°:  -46.7kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259921(US9512115, 25)copy SMILES
Affinity DataKi:  9.24nM ΔG°:  -46.6kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259904(US9512115, 7)copy SMILES
Affinity DataKi:  9.83nM ΔG°:  -46.5kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259917(US9512115, 21)copy SMILES
Affinity DataKi:  10.4nM ΔG°:  -46.3kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259904(US9512115, 7)copy SMILES
Affinity DataKi:  10.9nM ΔG°:  -46.2kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259921(US9512115, 25)copy SMILES
Affinity DataKi:  11.3nM ΔG°:  -46.1kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259920(US9512115, 24)copy SMILES
Affinity DataKi:  11.4nM ΔG°:  -46.1kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259926(US9512115, 30)copy SMILES
Affinity DataKi:  12.0nM ΔG°:  -46.0kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259926(US9512115, 30)copy SMILES
Affinity DataKi:  12.2nM ΔG°:  -45.9kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM98187(US8486940, 89 | US9650362, 89)copy SMILEScopy InChI
Affinity DataKi:  12.5nM IC50: 160nMAssay Description:Spectrophotometic Assay: This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spect...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2251GSFUS Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM98187(US8486940, 89 | US9650362, 89)copy SMILEScopy InChI
Affinity DataKi:  12.5nMAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometrical...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VD71H9US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259901(US9512115, 4)copy SMILES
Affinity DataKi:  12.6nM ΔG°:  -45.8kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259909(US9512115, 13)copy SMILES
Affinity DataKi:  13.1nM ΔG°:  -45.7kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259908(US9512115, 12)copy SMILES
Affinity DataKi:  13.1nM ΔG°:  -45.7kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259922(US9512115, 26)copy SMILES
Affinity DataKi:  13.6nM ΔG°:  -45.7kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM149371(US8962860, 16)copy SMILES
Affinity DataKi:  13.6nM ΔG°:  -45.7kJ/mole IC50: 128nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856V2US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259922(US9512115, 26)copy SMILES
Affinity DataKi:  14.3nM ΔG°:  -45.5kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259924(US9512115, 28)copy SMILES
Affinity DataKi:  14.9nM ΔG°:  -45.4kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM309890(1-(3,4,5- trimethoxyphenyl)-3- (3-(5-methyl-1H- im...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21Z46GVUS Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259918(US9512115, 22)copy SMILES
Affinity DataKi:  15.1nM ΔG°:  -45.4kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259923(US9512115, 27)copy SMILES
Affinity DataKi:  15.4nM ΔG°:  -45.3kJ/molepH: 6.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259908(US9512115, 12)copy SMILES
Affinity DataKi:  15.4nM ΔG°:  -45.3kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
PROBIODRUG AG

US Patent
LigandPNGBDBM259920(US9512115, 24)copy SMILES
Affinity DataKi:  15.5nM ΔG°:  -45.3kJ/molepH: 8.0 T: 2°CAssay Description:All measurements were performed with a BioAssay Reader HTS-7000Plus for microplates (Perkin Elmer) at 30° C. QC activity was evaluated fluorometr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DG4US Patent
Displayed 1 to 50 (of 550 total ) | Next | Last >>
Jump to: