TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2HD7X6XPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2HD7X6XPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 101nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 121nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 127nMAssay Description:Inhibition of c-MET (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 149nMAssay Description:Inhibition of wild type EGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Vichem Chemie Research Ltd.
Curated by ChEMBL
Vichem Chemie Research Ltd.
Curated by ChEMBL
Affinity DataIC50: 168nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair