Compile Data Set for Download or QSAR
Found 304 with Last Name = 'blake' and Initial = 'ra'
LigandPNGBDBM50448118(CHEMBL3122113 | US10590114, No. 80 | US11111235, N...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of LRRK2 G2019S mutant (unknown origin)More data for this Ligand-Target Pair
LigandPNGBDBM50398668(CHEMBL2178134 | US8802674, 256)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of LRRK2 G2019S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93N5PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50432188(CHEMBL2346976)copy SMILEScopy InChI
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of full length androgen receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93N5PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50432188(CHEMBL2346976)copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of androgen receptor LBD domain (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93N5PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523039(CHEMBL4591338)copy SMILEScopy InChI
Affinity DataIC50: 0.0100nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532101(CHEMBL4439408)copy SMILEScopy InChI
Affinity DataIC50: 0.0240nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T3WPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532101(CHEMBL4439408)copy SMILEScopy InChI
Affinity DataIC50: 0.0240nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T3WPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM368199((S)-2-(4-(2-(3-(fluoromethyl)azetidin-1-yl)ethoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.0300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM368199((S)-2-(4-(2-(3-(fluoromethyl)azetidin-1-yl)ethoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.0300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523049(CHEMBL4441471)copy SMILEScopy InChI
Affinity DataIC50: 0.0300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532103(CHEMBL4464224)copy SMILEScopy InChI
Affinity DataIC50: 0.0450nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523050(CHEMBL4455953)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572808(Gdc-9545 | Giredestrant | RO-7197597 | RO7197597)copy SMILES
Affinity DataIC50: 0.0500nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532105(CHEMBL4449709)copy SMILEScopy InChI
Affinity DataIC50: 0.0510nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T3WPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532102(CHEMBL4437985)copy SMILEScopy InChI
Affinity DataIC50: 0.0550nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532098(CHEMBL4464058)copy SMILEScopy InChI
Affinity DataIC50: 0.0590nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572809(CHEMBL4866043)copy SMILES
Affinity DataIC50: 0.0600nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523040(CHEMBL4463541)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572829(CHEMBL4856969)copy SMILES
Affinity DataIC50: 0.0700nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532106(CHEMBL4539802)copy SMILEScopy InChI
Affinity DataIC50: 0.0760nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T3WPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523035(CHEMBL4594150)copy SMILEScopy InChI
Affinity DataIC50: 0.0800nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572825(CHEMBL4856892)copy SMILES
Affinity DataIC50: 0.0800nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572826(CHEMBL4869698)copy SMILES
Affinity DataIC50: 0.0900nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572828(CHEMBL4864829)copy SMILES
Affinity DataIC50: 0.0900nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572832(CHEMBL4845726)copy SMILES
Affinity DataIC50: 0.0900nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM368199((S)-2-(4-(2-(3-(fluoromethyl)azetidin-1-yl)ethoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572821(CHEMBL4871161)copy SMILES
Affinity DataIC50: 0.100nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572824(CHEMBL4857736)copy SMILES
Affinity DataIC50: 0.130nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50542086(CHEMBL4649161)copy SMILEScopy InChI
Affinity DataIC50: 0.140nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572831(CHEMBL4877338)copy SMILES
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572823(CHEMBL4860671)copy SMILES
Affinity DataIC50: 0.160nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572834(CHEMBL4853118)copy SMILES
Affinity DataIC50: 0.160nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523057(CHEMBL4447143)copy SMILEScopy InChI
Affinity DataIC50: 0.170nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM299111(US10125135, Example 1)copy SMILES
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523053(CHEMBL4567402)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523054(CHEMBL4476031)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572822(CHEMBL4866232)copy SMILES
Affinity DataIC50: 0.230nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50238741(CHEBI:31638 | Faslodex | Fulvestrant | ICI-182780 ...)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572833(CHEMBL4873860)copy SMILES
Affinity DataIC50: 0.25nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523062(CHEMBL4450730)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50532104(CHEMBL1087419)copy SMILEScopy InChI
Affinity DataIC50: 0.280nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by Alexafluor-488 conjugate anti-mouse IgG antibody/Hoechst 33342 staining based imm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T3WPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572827(CHEMBL4871601)copy SMILES
Affinity DataIC50: 0.290nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572815(CHEMBL4847707)copy SMILES
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50508708(CHEMBL4438260)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523041(CHEMBL4588281)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572820(CHEMBL4850919)copy SMILES
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50572817(CHEMBL4854930)copy SMILES
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9T67PubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523051(CHEMBL4456532)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523042(CHEMBL4552853)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Genentech Inc.

Curated by ChEMBL
LigandPNGBDBM50523038(CHEMBL4470926)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by FITC/Hoechst 33342 staining based immunofluorescence imaging analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5M3VPubMed
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