Compile Data Set for Download or QSAR
Found 687 with Last Name = 'rampulla' and Initial = 'ra'
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi:  0.260nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541581(CHEMBL4646341)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541577(CHEMBL4646441)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541576(CHEMBL4644510)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541582(CHEMBL4636247)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541579(CHEMBL4637480)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541578(CHEMBL4638837)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition of human activated protein C using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541580(CHEMBL4639313)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541583(CHEMBL4633639)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541585(CHEMBL4635155)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267028(CHEMBL4073525)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Agonist activity at human GPR40 expressed in CHO-A12 cells assessed as increase in intracellular calcium flux measured for 100 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267031(CHEMBL4079930)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Agonist activity at human GPR40 expressed in CHO-A12 cells assessed as increase in intracellular calcium flux measured for 100 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541584(CHEMBL4639498)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Inhibition of human factor11a using pyro-Glu-Pro-Arg-pNA(para-nitroaniline) substrate by spectrophotometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetChymotrypsinogen B2(Homo sapiens)
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of human chymotrypsin by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267009(CHEMBL4089171)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267029(CHEMBL4069191)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267010(CHEMBL4082395)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267117(CHEMBL4060499)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267030(CHEMBL4090240)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267044(CHEMBL4069764)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267039(CHEMBL4090766)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267049(CHEMBL4095599)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Agonist activity at human GPR40 expressed in CHO-A12 cells assessed as increase in intracellular calcium flux measured for 100 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267035(CHEMBL4071899)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267038(CHEMBL4061093)copy SMILEScopy InChI
Affinity DataKi:  360nMAssay Description:Agonist activity at human GPR40 expressed in CHO-A12 cells assessed as increase in intracellular calcium flux measured for 100 secs by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267046(CHEMBL4103729)copy SMILEScopy InChI
Affinity DataKi:  890nMAssay Description:Agonist activity at human GPR40 expressed in CHO-A12 cells assessed as increase in intracellular calcium flux measured for 100 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267066(CHEMBL4067052)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267118(CHEMBL4096887)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetCoagulation factor XII(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of human factor-12a using H-(D)-CHT-Gly-ArgpNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267059(CHEMBL4091552)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of human factor-7a using H-(D)-Ile-Pro-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi:  4.10E+3nMAssay Description:Inhibition of human tissue-type plasminogen activator using methyl-sulfonyl-D-cyclohexylalanyl-Gly-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267047(CHEMBL4078852)copy SMILEScopy InChI
Affinity DataKi:  4.40E+3nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human plasma kallikrein using H-(D)-Pro-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267064(CHEMBL4070703)copy SMILEScopy InChI
Affinity DataKi:  6.50E+3nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >9.00E+3nMAssay Description:Inhibition of human factor-10a using N-benzoyl-Ile-Glu-(OH,OMe)-Gly-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267045(CHEMBL4063889)copy SMILEScopy InChI
Affinity DataKi:  9.00E+3nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetProthrombin(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >1.30E+4nMAssay Description:Inhibition of human thrombin using pyro-Glu-Pro-Arg-pNA(para-nitroaniline substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of human urokinase using pyro-Glu-Gly-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of human tissue-type plasminogen activator using H-(D)-Val-Leu-Lys-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetPlasminogen(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >2.10E+4nMAssay Description:Inhibition of human plasmin using H-(D)-Val-Leu-Lys-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267048(CHEMBL4075190)copy SMILEScopy InChI
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267021(CHEMBL4091669)copy SMILEScopy InChI
Affinity DataKi: >2.50E+4nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >2.70E+4nMAssay Description:Inhibition of human factor-9a using Methyl-sulfonyl-D-cyclohexylglycyl-Gly-Arg-AMC substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetKallikrein-1(Homo sapiens (Human))
Bristol Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50541586(CHEMBL4638245)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Inhibition of human tissue kallikrein-1 by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67MHGPubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50267113(CHEMBL4105565)copy SMILEScopy InChI
Affinity DataKi: >3.30E+4nMAssay Description:Binding affinity to human GPR40 expressed in HEK293 cell membranes after 1 hr by radioligand displacement based scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CD5PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50239718(CHEMBL4064666 | US10214537, Example 639)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7KVJPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50232433(CHEMBL4068514 | US10214537, Example 619)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7KVJPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Bristol-Myers Squibb Company

Curated by ChEMBL
LigandPNGBDBM50168472(CHEMBL3805348 | US9765060, Compound X)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Antisecretory activity evaluated by the inhibition of 14C -AP uptake in isolated rabbit parietal cells stimulated by exogenous histamineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7KVJPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center

Curated by ChEMBL
LigandPNGBDBM50544198(CHEMBL4636136)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542S4MPubMed
Displayed 1 to 50 (of 687 total ) | Next | Last >>
Jump to: