Compile Data Set for Download or QSAR
Found 214 with Last Name = 'laprairie' and Initial = 'rb'
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50556532(CHEMBL4753891)copy SMILES
Affinity DataKi:  0.790nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50601131(CHEMBL5193398)copy SMILES
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50601132(CHEMBL5204176)copy SMILES
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519776(CHEMBL4467516)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519778(CHEMBL4519310)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)copy SMILEScopy InChI
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50556532(CHEMBL4753891)copy SMILES
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid scintillation spectrometry ana...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50570253(CHEMBL4467500)copy SMILES
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)copy SMILEScopy InChI
Affinity DataKi:  34nMMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50586724(CHEMBL5082666)copy SMILES
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid scintillation spectrometry ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5S30PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519776(CHEMBL4467516)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519778(CHEMBL4519310)copy SMILEScopy InChI
Affinity DataKi:  94nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519795(CHEMBL4549068)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50517072(CHEMBL4450922)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membranes incubated for 60 mins by liquid scintillation spectrometry ana...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5S30PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50517072(CHEMBL4450922)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Displacement of [3H]CP55940 from human CB1R receptor expressed in CHO cell membranes after 60 mins by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50517072(CHEMBL4450922)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519795(CHEMBL4549068)copy SMILEScopy InChI
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]SR141716A from human CB1R receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50601132(CHEMBL5204176)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50570253(CHEMBL4467500)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50601131(CHEMBL5193398)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9PB9PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50023629(CHEMBL3341861)copy SMILEScopy InChI
Affinity DataEC50:  71nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500799(CHEMBL3758877)copy SMILEScopy InChI
Affinity DataEC50:  174nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Dalhousie University

Curated by ChEMBL
LigandPNGBDBM50500799(CHEMBL3758877)copy SMILEScopy InChI
Affinity DataEC50:  27nMAssay Description:Activity at CB1R in mouse brain membranes assessed as inhibition of CP55,940-induced [35S]GTPgammaS binding preincubated for 60 mins prior to [35S]GT...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500799(CHEMBL3758877)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Positive allosteric modulator activity at human CB1R expressed in CHO cells assessed as enhanced binding of [3H]CP55,940 after 60 mins by liquid scin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50389939(CHEMBL1553629)copy SMILEScopy InChI
Affinity DataEC50:  324nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)copy SMILEScopy InChI
Affinity DataEC50:  4.90nMAssay Description:Positive allosteric modulator activity at human CB1R expressed in CHO cells assessed as enhanced binding of [3H]CP55,940 after 60 mins by liquid scin...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500800(CHEMBL3758973)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500801(CHEMBL3758325)copy SMILEScopy InChI
Affinity DataEC50:  166nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500802(CHEMBL3758782)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500803(CHEMBL3758424)copy SMILEScopy InChI
Affinity DataEC50:  1.12E+3nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500804(CHEMBL3758817)copy SMILEScopy InChI
Affinity DataEC50:  389nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500800(CHEMBL3758973)copy SMILEScopy InChI
Affinity DataEC50:  683nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500805(CHEMBL3759542)copy SMILEScopy InChI
Affinity DataEC50:  43nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500801(CHEMBL3758325)copy SMILEScopy InChI
Affinity DataEC50:  28nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50023629(CHEMBL3341861)copy SMILEScopy InChI
Affinity DataEC50:  3.80nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500803(CHEMBL3758424)copy SMILEScopy InChI
Affinity DataEC50:  64nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500799(CHEMBL3758877)copy SMILEScopy InChI
Affinity DataEC50:  2.10nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500804(CHEMBL3758817)copy SMILEScopy InChI
Affinity DataEC50:  28nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50389939(CHEMBL1553629)copy SMILEScopy InChI
Affinity DataEC50:  9.10nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500805(CHEMBL3759542)copy SMILEScopy InChI
Affinity DataEC50:  118nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as effect on CP55,940-induced inhibition of forskolin-induced...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50389939(CHEMBL1553629)copy SMILEScopy InChI
Affinity DataEC50:  83nMAssay Description:Positive allosteric modulator activity at human CB1R expressed in CHO cells assessed as enhanced binding of [3H]CP55,940 after 60 mins by liquid scin...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50500802(CHEMBL3758782)copy SMILEScopy InChI
Affinity DataEC50:  209nMAssay Description:Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03C57PubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519774(CHEMBL4470555)copy SMILEScopy InChI
Affinity DataEC50:  700nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519775(CHEMBL4460580)copy SMILEScopy InChI
Affinity DataEC50:  43nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-stimu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519776(CHEMBL4467516)copy SMILEScopy InChI
Affinity DataEC50:  750nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519777(CHEMBL4469368)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced beta-arrestin2 recruitment af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50519778(CHEMBL4519310)copy SMILEScopy InChI
Affinity DataEC50:  26nMAssay Description:Allosteric agonist activity at N-terminal GFP-tagged rat CB1R expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50519776(CHEMBL4467516)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Positive allosteric modulatory activity at N-terminal GFP-tagged rat CB1R receptor expressed in HEK293 cells assessed as CP55940 EC50 for inhibition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50519778(CHEMBL4519310)copy SMILEScopy InChI
Affinity DataEC50:  1.70nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as increase in CP55940-induced inhibition of forskolin-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49GQPubMed
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