Affinity DataIC50: 4.40nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 202nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 206nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 233nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 325nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 417nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+3nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+3nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.43E+3nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 2.98E+3nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Tested in vitro for the HMG-CoA reductase inhibitory activity in a microsomal preparationMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+4nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 3.60E+4nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 5.10E+4nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 5.60E+4nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+4nMAssay Description:Compound was tested for inhibitory activity against squalene synthase using rat liver microsomal assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 1.20E+5nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1,/2,/3,/4, mitochondrial(Homo sapiens (Human))
Novartis Institute for Biomedical Research
Curated by ChEMBL
Novartis Institute for Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 2.00E+6nMAssay Description:In vitro inhibitory activity against pyruvate dehydrogenase kinase was determinedMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activity against PPAR-alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activity against PPAR-deltaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activity against PPAR-alphaMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Rattus norvegicus)
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Novartis Institutes for Biomedical Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Activity against PPAR-alphaMore data for this Ligand-Target Pair
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