Compile Data Set for Download or QSAR
Found 232 with Last Name = 'cox' and Initial = 'rf'
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM21363(12-chloro-9-(2-fluorophenyl)-3-methyl-2,4,8-triaza...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120343(3-[(S)-8-Chloro-6-(2-fluoro-phenyl)-2-methyl-4H-3,...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120340(3-[(S)-7-Chloro-5-(2-fluoro-phenyl)-2-oxo-2,3-dihy...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120353(3-[(S)-8-Chloro-6-(2-fluoro-phenyl)-4H-3,5,10b-tri...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120360(3-[(S)-8-Chloro-6-(2-fluoro-phenyl)-1-methyl-4H-3,...)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120344(3-[(S)-8-Chloro-6-(2-fluoro-phenyl)-1-methyl-4H-2,...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120359(3-((S)-8-Chloro-2-methyl-6-pyridin-2-yl-4H-3,5,10b...)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120357(3-((S)-8-Chloro-6-pyridin-2-yl-4H-3,5,10b-triaza-b...)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120345(3-[(S)-7-Chloro-5-(2-fluoro-phenyl)-2-methylamino-...)copy SMILEScopy InChI
Affinity DataKi:  96nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120358(3-((S)-8-Chloro-1-methyl-6-pyridin-2-yl-4H-3,5,10b...)copy SMILEScopy InChI
Affinity DataKi:  98nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120354(3-((S)-8-Chloro-1,2-dimethyl-6-pyridin-2-yl-4H-3,5...)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120347(3-((S)-7-Chloro-2-oxo-5-pyridin-2-yl-2,3-dihydro-1...)copy SMILEScopy InChI
Affinity DataKi:  139nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120349(3-[(S)-7-Chloro-2-ethylamino-5-(2-fluoro-phenyl)-3...)copy SMILEScopy InChI
Affinity DataKi:  146nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120352(3-{(S)-7-Chloro-5-(2-fluoro-phenyl)-2-[2-(1H-imida...)copy SMILEScopy InChI
Affinity DataKi:  208nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120351(3-[(S)-7-Chloro-5-(2-fluoro-phenyl)-2-(2-hydroxy-e...)copy SMILEScopy InChI
Affinity DataKi:  303nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50007664(7-chloro-2-methylamino-5-phenyl-3H-1,4-benzodiazep...)copy SMILEScopy InChI
Affinity DataKi:  438nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120355(3-[(S)-7-Chloro-5-(2-fluoro-phenyl)-2-(2-pyridin-4...)copy SMILEScopy InChI
Affinity DataKi:  792nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120350(3-[(S)-2-Benzylamino-7-chloro-5-(2-fluoro-phenyl)-...)copy SMILEScopy InChI
Affinity DataKi:  875nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120348(3-[(S)-7-Chloro-5-(2-fluoro-phenyl)-2-isobutylamin...)copy SMILEScopy InChI
Affinity DataKi:  1.01E+3nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120361(3-((S)-7-Chloro-2-methylamino-5-pyridin-2-yl-3H-be...)copy SMILEScopy InChI
Affinity DataKi:  1.08E+3nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120356(3-{(S)-7-Chloro-5-(2-fluoro-phenyl)-2-[(pyridin-4-...)copy SMILEScopy InChI
Affinity DataKi:  1.23E+3nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetTranslocator protein(Rattus norvegicus (rat))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50120346(3-[(R)-8-Chloro-6-(2-fluoro-phenyl)-1-methyl-4H-2,...)copy SMILEScopy InChI
Affinity DataKi:  3.57E+3nMAssay Description:Binding affinity of the compound was determined against rat benzodiazepine (BZD) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ6X4FPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271750(CHEMBL4126095)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271775(CHEMBL4129590)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271748(CHEMBL4128577)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271747(CHEMBL4127245)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271734(CHEMBL4128540)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271738(CHEMBL4129219)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50296011(2-cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271780(CHEMBL4126511)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
LigandPNGBDBM50271756(CHEMBL4127319)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of PI3Kgamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271752(CHEMBL4128114)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271739(CHEMBL4126740)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271728(CHEMBL4127977)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271751(CHEMBL4127140)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271744(CHEMBL4128939)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271774(CHEMBL4128459)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271788(CHEMBL4127064)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271740(CHEMBL4127330)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271729(CHEMBL4128717)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271741(CHEMBL4129791)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271777(CHEMBL4129362)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271755(CHEMBL4129843)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50296009(2-ethyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271778(CHEMBL4130310)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271745(CHEMBL4126566)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50296010(2-isobutyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271776(CHEMBL4125907)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271779(CHEMBL4127479)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of full-length human GST-tagged CAMKK2 using 5FAM-AKPKGNKDYHLQTCCGSLAYRRR-amide as substrate preincubated for 30 mins followed by substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50271740(CHEMBL4127330)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of CAMKK2 in mouse N39 cells assessed as decrease in AMPKalpha phosphorylation at T172 preincubated for 80 mins followed by inomycin addit...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DFBPubMed
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