Compile Data Set for Download or QSAR
Found 5 with Last Name = 'jenkins' and Initial = 'rg'
LigandPNGBDBM50287709((E)-3-Carboxy-2-(16-sulfooxy-hexadecyl)-pent-2-ene...)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:In vitro inhibition of human recombinant Protein farnesyltransferase with respect to FPPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TQ1
LigandPNGBDBM50287707((E)-3-Carboxy-2-(16-hydroxy-hexadecyl)-pent-2-ened...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:In vitro inhibition of human recombinant Protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TQ1
LigandPNGBDBM50287708((E)-3-Methoxycarbonyl-2-(16-sulfooxy-hexadecyl)-pe...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of human recombinant Protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TQ1
LigandPNGBDBM50287709((E)-3-Carboxy-2-(16-sulfooxy-hexadecyl)-pent-2-ene...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of human recombinant Protein farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2222TQ1
LigandPNGBDBM50478520(BARCELONEIC ACID A)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human recombinant FPTase by Ras farnesyl-protein-transferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6V1WPubMed