Compile Data Set for Download or QSAR
Found 120 with Last Name = 'walker' and Initial = 'rg'
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552190(CHEMBL4741714)copy SMILES
Affinity DataIC50: 0.00600nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))TBA
LigandPNGBDBM50552190(CHEMBL4741714)copy SMILES
Affinity DataIC50: 0.00900nMAssay Description:Inhibition of PIM3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))TBA
LigandPNGBDBM50552190(CHEMBL4741714)copy SMILES
Affinity DataIC50: 0.0180nMAssay Description:Inhibition of PIM2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50387298(CHEMBL2048872)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human PIM1 using full-length BAD as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552189(CHEMBL4793492)copy SMILES
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human PIM1 using full length BAD peptide substrate in presence of ATP at Km concentrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248903(CHEMBL4060012)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))TBA
LigandPNGBDBM50387298(CHEMBL2048872)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PIM3 using full-length BAD as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))TBA
LigandPNGBDBM50552189(CHEMBL4793492)copy SMILES
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PIM3 using full length BAD peptide substrate in presence of ATP at Km concentrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248920(CHEMBL4079975)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248897(CHEMBL4061984)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248893(CHEMBL4104431)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248921(CHEMBL4096030)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552147(CHEMBL4794742)copy SMILES
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50436459(CHEMBL2396661)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of P13Kalpha (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50387298(CHEMBL2048872)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human PIM2 using full-length BAD as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248898(CHEMBL4083726)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))TBA
LigandPNGBDBM50552189(CHEMBL4793492)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of human PIM2 using full length BAD peptide substrate in presence of ATP at Km concentrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552146(CHEMBL4747343)copy SMILES
Affinity DataIC50: 5.20nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248863(CHEMBL4087322)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248904(CHEMBL4069560)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248892(CHEMBL4074078)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552149(CHEMBL4778893)copy SMILES
Affinity DataIC50: 6.90nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248894(CHEMBL4060062)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50364776(CHEMBL1952141 | CHEMBL1952329)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human full length N-terminal GST-tagged PIM1 expressed in Escherichia coli using KKRNRTLTV as substrate incubated for 40 mi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50364776(CHEMBL1952141 | CHEMBL1952329)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human full length N-terminal GST-tagged PIM1 expressed in Escherichia coli using LKKRNRTLTV as substrate measured after 40 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248899(CHEMBL4069566)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552171(CHEMBL4757567)copy SMILES
Affinity DataIC50: 9nMAssay Description:Inhibition of human PIM1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248860(CHEMBL4077499)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552173(CHEMBL4788212)copy SMILES
Affinity DataIC50: 11nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248901(CHEMBL4075979)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248922(CHEMBL4077328)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552150(CHEMBL4797284)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552153(CHEMBL4794863)copy SMILES
Affinity DataIC50: 15nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552155(CHEMBL4777003)copy SMILES
Affinity DataIC50: 15nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248923(CHEMBL4075290)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552154(CHEMBL4798741)copy SMILES
Affinity DataIC50: 18nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552178(CHEMBL4758677)copy SMILES
Affinity DataIC50: 20nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248900(CHEMBL4075977)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552171(CHEMBL4757567)copy SMILES
Affinity DataIC50: 22nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552157(CHEMBL4786077)copy SMILES
Affinity DataIC50: 22nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552163(CHEMBL4783270)copy SMILES
Affinity DataIC50: 24nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248864(CHEMBL4090574)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248895(CHEMBL4088298)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552152(CHEMBL4783323)copy SMILES
Affinity DataIC50: 28nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552184(CHEMBL4751389)copy SMILES
Affinity DataIC50: 33nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248865(CHEMBL4069055)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50248896(CHEMBL4068718)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant PIM1 (unknown origin) by pyruvate kinase/lactate dehydrogenase-coupled assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M5VPubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552185(CHEMBL4781049)copy SMILES
Affinity DataIC50: 37nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552151(CHEMBL4763088)copy SMILES
Affinity DataIC50: 40nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))TBA
LigandPNGBDBM50552172(CHEMBL4742215)copy SMILES
Affinity DataIC50: 40nMAssay Description:Inhibition of PIM1 (unknown origin) by coupled kinetic assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3607PubMed
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