Compile Data Set for Download or QSAR
Found 17 with Last Name = 'pipitone' and Initial = 'rm'
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant HDAC1 using modified Boc-Lys(Ac)-AMC MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026643(CHEMBL3335369)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of human recombinant HDAC1 using modified Boc-Lys(Ac)-AMC MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026641(CHEMBL3335367)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of human recombinant HDAC1 using modified Boc-Lys(Ac)-AMC MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50135180(CHEMBL3746143)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN97GZPubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026643(CHEMBL3335369)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human recombinant HDAC6 using Z-MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026644(CHEMBL3335370)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant HDAC6 using Z-MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50135175(CHEMBL490384)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN97GZPubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50135177(CHEMBL3747558)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN97GZPubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026644(CHEMBL3335370)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant HDAC1 using modified Boc-Lys(Ac)-AMC MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human recombinant HDAC6 using Z-MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMedDrugBank
TargetHistone deacetylase 4(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026644(CHEMBL3335370)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human recombinant HDAC4 using (S)-[5-Acetylamino-1-(2-oxo-4-trifluorometyl-2Hchromen-7-ylcarbamoyl)pentl]carbami acid tert-Butyl Ester ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of human recombinant HDAC4 using (S)-[5-Acetylamino-1-(2-oxo-4-trifluorometyl-2Hchromen-7-ylcarbamoyl)pentl]carbami acid tert-Butyl Ester ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026642(CHEMBL3335368)copy SMILEScopy InChI
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human recombinant HDAC1 using modified Boc-Lys(Ac)-AMC MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026643(CHEMBL3335369)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of human recombinant HDAC4 using (S)-[5-Acetylamino-1-(2-oxo-4-trifluorometyl-2Hchromen-7-ylcarbamoyl)pentl]carbami acid tert-Butyl Ester ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026629(CHEMBL3334509)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of human recombinant HDAC1 using modified Boc-Lys(Ac)-AMC MAL as substrate after 1 hr by fluorescent activity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V70PubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50135176(CHEMBL3747491)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of bovine brain tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN97GZPubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£ di Ferrara

Curated by ChEMBL
LigandPNGBDBM50135178(CHEMBL3745749)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of bovine brain tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN97GZPubMed