Compile Data Set for Download or QSAR
Found 195 with Last Name = 'law' and Initial = 'rp'
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189403(CHEMBL3828191)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of full length BRPF1 in human HUT78 cell nuclear/chromatin extract after 45 mins by chemoproteomic competition binding assayMore data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189392(CHEMBL3828311)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50028142(CHEMBL2177300)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189403(CHEMBL3828191)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50028142(CHEMBL2177300)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y390A mutant BD1 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189402(CHEMBL3828008)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189403(CHEMBL3828191)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Binding affinity to NanoLuc-tagged BRPF1 isoform 1 bromodomain (625 to 735 residues) (unknown origin) expressed in HEK293 cells co-transfected with h...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189353(CHEMBL3827767)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455493(CHEMBL4213809)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of BRD3 BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189409(CHEMBL3828684)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y390A mutant BD1 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50032927(CHEMBL3356143 | N-[2,3-Dihydro-1,3-dimethyl-2-oxo-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189408(CHEMBL3828194)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455492(CHEMBL4211868)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455490(CHEMBL4205865)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455493(CHEMBL4213809)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of BRD3 BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455508(CHEMBL4205557)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455500(CHEMBL4207924)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189348(CHEMBL3827114)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455507(CHEMBL4212836)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189357(CHEMBL3827560)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189405(CHEMBL3828354)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189411(CHEMBL3827996)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455479(CHEMBL4217789)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455484(CHEMBL4208455)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455493(CHEMBL4213809)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human BRD2 BD2 after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189354(CHEMBL3828061)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189339(CHEMBL3828500)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189340(CHEMBL3828146)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455493(CHEMBL4213809)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of BRDT BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455482(CHEMBL4213381)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189410(CHEMBL3828449)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50032928(CHEMBL3356145)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189406(CHEMBL3827280)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455501(CHEMBL4216840)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189351(CHEMBL3827276)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189404(CHEMBL3828026)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455491(CHEMBL4208993)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455510(CHEMBL4204112)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455511(CHEMBL4218207)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455512(CHEMBL4206478)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189338(CHEMBL3828399)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetPeregrin(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50189381(CHEMBL3828504)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Esc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S184G2PubMed
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of BRDT BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455482(CHEMBL4213381)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y390A mutant BD1 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455506(CHEMBL4208636)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Displacement of (+)-JQ1 from 6H-Thr BRD4 Y97A mutant BD2 (unknown origin) after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
TargetBromodomain-containing protein 2(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50455480(CHEMBL4218735)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Inhibition of human BRD2 BD2 after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1N6WPubMed
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