Compile Data Set for Download or QSAR
Found 480 with Last Name = 'cesarini' and Initial = 's'
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X069TRPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MHGPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against HIV-1 wild type reverse transcriptase (IIIB)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (Y181C)More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of HIV1 virion-associated reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56NJRPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168052((4-Iodo-phenyl)-thiocarbamic acid 2-(1,3-dioxo-1,3...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibitory concentration against HIV-1 wild type reverse transcriptase (IIIB)More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50480227(CHEMBL520032)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X069TRPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103N+Y181C)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168128(CHEMBL191655 | O-2-(1,3-dioxoisoindolin-2-yl)ethyl...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibitory concentration against HIV-1 virion reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50480228(CHEMBL484982)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of wild-type HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X069TRPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50478732(CHEMBL443403)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Inhibition of HIV1 virion-associated reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56NJRPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50478749(CHEMBL471541)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MHGPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM1866(3-(5-bromopyridin-2-yl)-1-[2-(pyridin-2-yl)ethyl]t...)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MHGPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM1866(3-(5-bromopyridin-2-yl)-1-[2-(pyridin-2-yl)ethyl]t...)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibitory concentration against HIV-1 wild type reverse transcriptase (IIIB)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM1866(3-(5-bromopyridin-2-yl)-1-[2-(pyridin-2-yl)ethyl]t...)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of HIV1 virion-associated reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56NJRPubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50478750(CHEMBL471691)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of HIV1 recombinant wild type reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MHGPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168060(CHEMBL195108 | N-[2-(4-Iodo-phenylthiocarbamoyloxy...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory concentration against HIV-1 wild type reverse transcriptase (IIIB)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103R)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168052((4-Iodo-phenyl)-thiocarbamic acid 2-(1,3-dioxo-1,3...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103R)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168060(CHEMBL195108 | N-[2-(4-Iodo-phenylthiocarbamoyloxy...)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (Y181C)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM1866(3-(5-bromopyridin-2-yl)-1-[2-(pyridin-2-yl)ethyl]t...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (Y181C)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168052((4-Iodo-phenyl)-thiocarbamic acid 2-(1,3-dioxo-1,3...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (Y181C)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168052((4-Iodo-phenyl)-thiocarbamic acid 2-(1,3-dioxo-1,3...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103N+Y181C)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM1866(3-(5-bromopyridin-2-yl)-1-[2-(pyridin-2-yl)ethyl]t...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103R)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM1866(3-(5-bromopyridin-2-yl)-1-[2-(pyridin-2-yl)ethyl]t...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103N+Y181C)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168060(CHEMBL195108 | N-[2-(4-Iodo-phenylthiocarbamoyloxy...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103N+Y181C)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Universit£ di Genova

Curated by ChEMBL
LigandPNGBDBM50168060(CHEMBL195108 | N-[2-(4-Iodo-phenylthiocarbamoyloxy...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against HIV-1 mutant reverse transcriptase (K103R)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JQKPubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
Laboratoire de Chimie et de Biochimie Pharmacologiques et Toxicologiques , CNRS UMR 8601, Université Paris Descartes, Sorbonne Paris Cité , 45 rue des Saints-Pères , 75270 Paris Cedex 06 , France.

Curated by ChEMBL
LigandPNGBDBM50446782(CHEMBL3114672)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+6nMAssay Description:Antagonist activity at rat GluN1a/GluN2A receptors expressed in Xenopus laevis oocytes assessed as inhibition of L-glutamate/glucine induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0BR0PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(RAT)
Laboratoire de Chimie et de Biochimie Pharmacologiques et Toxicologiques , CNRS UMR 8601, Université Paris Descartes, Sorbonne Paris Cité , 45 rue des Saints-Pères , 75270 Paris Cedex 06 , France.

Curated by ChEMBL
LigandPNGBDBM50446782(CHEMBL3114672)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+6nMAssay Description:Antagonist activity at rat GluN1a/mouse GluN2B receptors expressed in Xenopus laevis oocytes assessed as inhibition of L-glutamate/glucine induced cu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0BR0PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM82006(D-AP4 | D-APB | US9212196, L-AP4)copy SMILEScopy InChI
Affinity DataEC50:  130nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196906(US9212196, Derivative 2)copy SMILEScopy InChI
Affinity DataEC50:  110nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196907(US9212196, Derivative 3)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196908(US9212196, Derivative 4)copy SMILEScopy InChI
Affinity DataEC50:  500nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196909(US9212196, Derivative 5)copy SMILEScopy InChI
Affinity DataEC50:  280nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196910(US9212196, Derivative 6)copy SMILEScopy InChI
Affinity DataEC50:  80nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196911(US9212196, Derivative 7)copy SMILEScopy InChI
Affinity DataEC50:  130nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196912(US9212196, Derivative 8)copy SMILEScopy InChI
Affinity DataEC50:  150nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196913(US9212196, Derivative 9)copy SMILEScopy InChI
Affinity DataEC50:  380nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196914(US9212196, Derivative 10)copy SMILEScopy InChI
Affinity DataEC50:  530nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196915(US9212196, Derivative 11)copy SMILEScopy InChI
Affinity DataEC50:  480nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196916(US9212196, Derivative 12)copy SMILEScopy InChI
Affinity DataEC50:  980nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196917(US9212196, Derivative 13)copy SMILEScopy InChI
Affinity DataEC50:  1.22E+4nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196918(US9212196, Derivative 14)copy SMILEScopy InChI
Affinity DataEC50:  370nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196919(US9212196, Derivative 15)copy SMILEScopy InChI
Affinity DataEC50:  7.60E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196920(US9212196, Derivative 16 | US9212196, Derivative 1...)copy SMILEScopy InChI
Affinity DataEC50:  4.90E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196920(US9212196, Derivative 16 | US9212196, Derivative 1...)copy SMILEScopy InChI
Affinity DataEC50:  1.30E+4nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196922(US9212196, Derivative 18)copy SMILEScopy InChI
Affinity DataEC50:  2.50E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196923(US9212196, Derivative 19)copy SMILEScopy InChI
Affinity DataEC50:  1.67E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196924(US9212196, Derivative 20)copy SMILEScopy InChI
Affinity DataEC50:  60nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196925(US9212196, Derivative 21)copy SMILEScopy InChI
Affinity DataEC50:  900nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
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