Compile Data Set for Download or QSAR
Found 112 with Last Name = 'heinzlmeir' and Initial = 's'
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50299218(8-(2-Methoxyphenyl)-1-methyl-7-(2'-methyl-5'-hydro...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9W5MPubMed
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM209859(4-N-(5-cyclopropyl-1H-pyrazol-3-yl)-6-(4-methylpip...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9W5MPubMed
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50311316(CHEMBL1077739 | LDN-211904 | N-(2-chlorophenyl)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM209858(Danusertib | N-[5-[(2R)-2-methoxy-2-phenylacetyl]-...)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM209861(5-(3-ethylsulfonylphenyl)-3,8-dimethyl-N-(1-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 4.80nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9W5MPubMed
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM6568(6-(2,6-dichlorophenyl)-8-methyl-2-{[3-(methylsulfa...)copy SMILEScopy InChI
Affinity DataIC50: 7.90nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50100615(E-7050 | E7050 | Golvatinib)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM209860(4-[[(3S)-3-(dimethylamino)pyrrolidin-1-yl]methyl]-...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9W5MPubMed
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50382959(CEP-32496 | CHEMBL2029988 | US9730937, Example 261)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9W5MPubMed
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50237710(4-methyl-N-[3-(4-methyl-1H-imidazol-1-yl)-5-(trifl...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9W5MPubMed
TargetEphrin type-A receptor 2 [596-900](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50277545(4-(9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Refer to Reaction Biology Corps.More data for this Ligand-Target Pair
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601516(CHEMBL5181586)copy SMILES
Affinity DataIC50: 80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601516(CHEMBL5181586)copy SMILES
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601515(CHEMBL5194499)copy SMILES
Affinity DataIC50: 310nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601518(CHEMBL5173110)copy SMILES
Affinity DataIC50: 740nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601530(CHEMBL5203844)copy SMILES
Affinity DataIC50: 850nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601532(CHEMBL5186486)copy SMILES
Affinity DataIC50: 990nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601517(CHEMBL5181611)copy SMILES
Affinity DataIC50: 990nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601529(CHEMBL5176431)copy SMILES
Affinity DataIC50: 1.05E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601530(CHEMBL5203844)copy SMILES
Affinity DataIC50: 1.18E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601527(CHEMBL5178796)copy SMILES
Affinity DataIC50: 1.22E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601531(CHEMBL5184488)copy SMILES
Affinity DataIC50: 1.54E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601532(CHEMBL5186486)copy SMILES
Affinity DataIC50: 1.59E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601515(CHEMBL5194499)copy SMILES
Affinity DataIC50: 1.85E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601521(CHEMBL5092273)copy SMILES
Affinity DataIC50: 2.15E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601528(CHEMBL5176119)copy SMILES
Affinity DataIC50: 2.87E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601524(CHEMBL5201006)copy SMILES
Affinity DataIC50: 2.99E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601520(CHEMBL5185035)copy SMILES
Affinity DataIC50: 3.29E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601519(CHEMBL5191015)copy SMILES
Affinity DataIC50: 3.93E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601527(CHEMBL5178796)copy SMILES
Affinity DataIC50: 4.18E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601517(CHEMBL5181611)copy SMILES
Affinity DataIC50: 4.30E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601529(CHEMBL5176431)copy SMILES
Affinity DataIC50: 4.92E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601522(CHEMBL5186307)copy SMILES
Affinity DataIC50: 4.95E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601533(CHEMBL5171029)copy SMILES
Affinity DataIC50: 5.21E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601518(CHEMBL5173110)copy SMILES
Affinity DataIC50: 8.65E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601531(CHEMBL5184488)copy SMILES
Affinity DataIC50: 1.25E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601521(CHEMBL5092273)copy SMILES
Affinity DataIC50: 1.36E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601528(CHEMBL5176119)copy SMILES
Affinity DataIC50: 1.41E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601523(CHEMBL5180413)copy SMILES
Affinity DataIC50: 1.58E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50601524(CHEMBL5201006)copy SMILES
Affinity DataIC50: 1.58E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20Z77B9PubMed
TargetFerrochelatase, mitochondrial [R115L](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM185145(7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-(3-phenylm...)copy SMILEScopy InChI
Affinity DataKd:  4.40E+3nMAssay Description:Briefly, 5 mg of a protein mixture of the four cell lines or a single cell line were incubated with compound dilution series in DMSO (3 nM, 10 nM, 30...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB51R8PubMed
TargetFerrochelatase, mitochondrial [R115L](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM185146(6-[5-[(2-methylsulfonylethylamino)methyl]furan-2-y...)copy SMILEScopy InChI
Affinity DataKd:  6.40E+3nMAssay Description:Briefly, 5 mg of a protein mixture of the four cell lines or a single cell line were incubated with compound dilution series in DMSO (3 nM, 10 nM, 30...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB51R8PubMed
TargetFerrochelatase, mitochondrial [R115L](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM25117(AG-013736 | AXITINIB | N-methyl-2-({3-[(E)-2-(pyri...)copy SMILEScopy InChI
Affinity DataKd:  3.10E+3nMAssay Description:Briefly, 5 mg of a protein mixture of the four cell lines or a single cell line were incubated with compound dilution series in DMSO (3 nM, 10 nM, 30...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB51R8PubMed
TargetFerrochelatase, mitochondrial [R115L](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50429701(AZD-2014 | CHEMBL2336325 | US9102670, 1ap)copy SMILEScopy InChI
Affinity DataKd:  3.40E+3nMAssay Description:Briefly, 5 mg of a protein mixture of the four cell lines or a single cell line were incubated with compound dilution series in DMSO (3 nM, 10 nM, 30...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB51R8PubMed
TargetFerrochelatase, mitochondrial [R115L](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50246253(4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)-N-(4-(me...)copy SMILEScopy InChI
Affinity DataKd:  2.60E+3nMAssay Description:Briefly, 5 mg of a protein mixture of the four cell lines or a single cell line were incubated with compound dilution series in DMSO (3 nM, 10 nM, 30...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB51R8PubMed
TargetFerrochelatase, mitochondrial [R115L](Homo sapiens (Human))
Technical University of Munich

LigandPNGBDBM50348452(AZD-8055 | CHEMBL1801204 | US9102670, 1a)copy SMILEScopy InChI
Affinity DataKd:  6.20E+3nMAssay Description:Briefly, 5 mg of a protein mixture of the four cell lines or a single cell line were incubated with compound dilution series in DMSO (3 nM, 10 nM, 30...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB51R8PubMed
Displayed 1 to 50 (of 112 total ) | Next | Last >>
Jump to: