Affinity DataKi: 0.390nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.870nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity against human Alpha-2A adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 166nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 189nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 843nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 990nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Binding affinity against human alpha 2b-adrenergic receptor expressed stably in CHO cells using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair