TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 127nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 276nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.13E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+3nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of 5-LO in A23187/AA-stimulated human intact neutrophils assessed as reduction in LTB4/5-HETE formation measured after 20 mins by RP-HPLC ...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of mPGES-1 obtained from IL-beta stimulated human A549 cells microsomes assessed as residual activity by measuring conversion of PGH2 to P...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 2.05E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 2.57E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 2.84E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 3.38E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 3.45E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
Affinity DataIC50: 4.04E+4nMAssay Description:Antagonist activity at human FXR transfected in HepG2 cells assessed as inhibition of CDCA-induced receptor transactivation by luciferase reporter as...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair
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