Compile Data Set for Download or QSAR
Found 91 with Last Name = 'orive' and Initial = 's'
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450436(CHEMBL4173663)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450440(CHEMBL4170829)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450437(CHEMBL4177037)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450439(CHEMBL4162307)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450289(CHEMBL4172928)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450435(CHEMBL4165748)copy SMILEScopy InChI
Affinity DataKi:  251nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450441(CHEMBL4173387)copy SMILEScopy InChI
Affinity DataKi:  251nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450438(CHEMBL4166818)copy SMILEScopy InChI
Affinity DataKi:  398nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450443(CHEMBL4174307)copy SMILEScopy InChI
Affinity DataKi:  794nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450434(CHEMBL4172349)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Ogeda SA

Curated by ChEMBL
LigandPNGBDBM50450442(CHEMBL4170872)copy SMILEScopy InChI
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]ES227703 from human FFA2R expressed in CHOK1 cells after 60 mins by TopCount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0R8RPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261349(CHEMBL4073785)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of DNA-PK in human HeLa nuclear extracts incubated for 40 mins using calf thymus DNA and fluoroscein-p53[Ser15]-peptide by Lanthascreen ti...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261349(CHEMBL4073785)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human DNA-PK catalytic subunit using DNA and [EPPLSQEAFADLWKK] peptide substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202255(CHEMBL3982304)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50426450(CHEMBL2322664)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of PI3Kbeta in human washed platelets assessed as suppression of ADP-induced platelet aggregation preincubated for 5 mins followed by ADP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202255(CHEMBL3982304)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of PI3Kbeta in human washed platelets assessed as suppression of ADP-induced platelet aggregation preincubated for 5 mins followed by ADP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50426459(CHEMBL2322668)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of PI3Kbeta in human washed platelets assessed as suppression of ADP-induced platelet aggregation preincubated for 5 mins followed by ADP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202255(CHEMBL3982304)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of human DNA-PK catalytic subunit using DNA and [EPPLSQEAFADLWKK] peptide substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50447094(CHEMBL1972466)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202259(CHEMBL3930788)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202264(CHEMBL3949883)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202254(CHEMBL3953591)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202259(CHEMBL3930788)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202279(CHEMBL3922132)copy SMILEScopy InChI
Affinity DataIC50: 428nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202265(CHEMBL3963433)copy SMILEScopy InChI
Affinity DataIC50: 521nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202252(CHEMBL3917147)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202263(CHEMBL3948855)copy SMILEScopy InChI
Affinity DataIC50: 554nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202256(CHEMBL3936124)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202253(CHEMBL3958556)copy SMILEScopy InChI
Affinity DataIC50: 811nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202266(CHEMBL3893326)copy SMILEScopy InChI
Affinity DataIC50: 955nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202264(CHEMBL3949883)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202288(CHEMBL3972268)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202252(CHEMBL3917147)copy SMILEScopy InChI
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202262(CHEMBL3978019)copy SMILEScopy InChI
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202258(CHEMBL3962354)copy SMILEScopy InChI
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202257(CHEMBL3974302)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202261(CHEMBL3908177)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202267(CHEMBL3900274)copy SMILEScopy InChI
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50261354(CHEMBL4103756)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50261337(CHEMBL4074385)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50261355(CHEMBL4071376)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261329(CHEMBL4077367)copy SMILEScopy InChI
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50426450(CHEMBL2322664)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of PI3Kbeta in human platelet-rich plasma assessed as suppression of ADP-induced platelet aggregation preincubated for 5 mins followed by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50261339(CHEMBL4079378)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50202268(CHEMBL3935927)copy SMILEScopy InChI
Affinity DataIC50: 2.84E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) expressed in Escherichia coli-infected fall armyworm sf21 cells co-expressing p85 by kinase-glo luminescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X59RNPubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50261347(CHEMBL4104565)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of wild type PI3K-delta (unknown origin) assessed as decrease in ATP consumption using phosphotidylinositol bisphosphate and ATP measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261350(CHEMBL4091681)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50261328(CHEMBL4083912)copy SMILEScopy InChI
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of human PDE3A by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XKGPubMed
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