TargetReverse transcriptase(Human immunodeficiency virus 1)
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of reverse transcriptase activity in HIV1 infected HeLa-MAGI cells at 37 deg C after 48 hrsMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of reverse transcriptase activity in HIV1 NL4-3 infected MT4 cells before dialysisMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of reverse transcriptase activity in HIV1 infected HeLa-MAGI cells at 37 deg C after 48 hrsMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of reverse transcriptase activity in HIV1 NL4-3 infected MT4 cells after dialysisMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
School of Pharmacy, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom.
Curated by ChEMBL
School of Pharmacy, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom.
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
School of Pharmacy, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom.
Curated by ChEMBL
School of Pharmacy, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom.
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Universidade Federal do Rio de Janeiro
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of reverse transcriptase activity in HIV1 NL4-3 infected MT4 cells before dialysisMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
School of Pharmacy, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom.
Curated by ChEMBL
School of Pharmacy, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, United Kingdom.
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human His-tagged LSD1 expressed in Escherichia coli BL21 (DE3) using H3K4me2 peptide as substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Irreversible inhibition of Trypanosoma cruzi cruzipainMore data for this Ligand-Target Pair
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