Compile Data Set for Download or QSAR
Found 65 with Last Name = 'piguel' and Initial = 's'
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University

Curated by ChEMBL
LigandPNGBDBM50466393(CHEMBL4277499)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50384576(CHEMBL2036808)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Inhibition of MER (unknown origin)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466394(CHEMBL4285809)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University

Curated by ChEMBL
LigandPNGBDBM50431281(CHEMBL2347987)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of AXL (unknown origin) phosphorylation expressed in mouse NIH/3T3 cells after 2 hrs by immunoprecipitation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University

Curated by ChEMBL
LigandPNGBDBM50384576(CHEMBL2036808)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466392(CHEMBL4285448)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50384576(CHEMBL2036808)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of TYRO3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM7576(1-(6-{[(4-chlorophenyl)methyl]amino}-9-(propan-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 60nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University

Curated by ChEMBL
LigandPNGBDBM50466392(CHEMBL4285448)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466393(CHEMBL4277499)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM7573(1-(6-{[(4-methoxyphenyl)methyl]amino}-9-(propan-2-...)copy SMILEScopy InChI
Affinity DataIC50: 230nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466394(CHEMBL4285809)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466393(CHEMBL4277499)copy SMILEScopy InChI
Affinity DataIC50: 690nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10651(2-purine deriv. 17 | 4-(6-{[(4-methoxyphenyl)methy...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10643(2-arylpurine deriv. 8 | 4-{6-[(2-methoxyethyl)amin...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10643(2-arylpurine deriv. 8 | 4-{6-[(2-methoxyethyl)amin...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10651(2-purine deriv. 17 | 4-(6-{[(4-methoxyphenyl)methy...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10646(2-arylpurine deriv. 11 | 4-{6-[(2-methoxyethyl)ami...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University

Curated by ChEMBL
LigandPNGBDBM50466394(CHEMBL4285809)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10650(2-purine deriv. 15 | 5-{6-[(2-methoxyethyl)amino]-...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10650(2-purine deriv. 15 | 5-{6-[(2-methoxyethyl)amino]-...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10645(2-arylpurine deriv. 10 | N-(4-{6-[(2-methoxyethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10644(1-(4-{6-[(2-methoxyethyl)amino]-9-(propan-2-yl)-9H...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10644(1-(4-{6-[(2-methoxyethyl)amino]-9-(propan-2-yl)-9H...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10645(2-arylpurine deriv. 10 | N-(4-{6-[(2-methoxyethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10646(2-arylpurine deriv. 11 | 4-{6-[(2-methoxyethyl)ami...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10649(1-(5-{6-[(2-methoxyethyl)amino]-9-(propan-2-yl)-9H...)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10647(2-arylpurine deriv. 12 | N-(2-cyanoethyl)-4-{6-[(2...)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10648(2-arylpurine deriv. 13 | methyl N-(4-{6-[(2-methox...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10647(2-arylpurine deriv. 12 | N-(2-cyanoethyl)-4-{6-[(2...)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetCyclin-dependent kinase 1/G2/mitotic-specific cyclin-B(Marthasterias glacialis (starfish))
Institut Curie

LigandPNGBDBM10648(2-arylpurine deriv. 13 | methyl N-(4-{6-[(2-methox...)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466392(CHEMBL4285448)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetCyclin-dependent kinase 5 activator 1 [99-307](Homo sapiens (Human))
Institut Curie

LigandPNGBDBM10649(1-(5-{6-[(2-methoxyethyl)amino]-9-(propan-2-yl)-9H...)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+3nMpH: 7.2 T: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50113707(2,6,9-Trisubstitute purine, 2 | 2-(2-hydroxyethyla...)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of MER (588 to 855) (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466391(CHEMBL4293688)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50466391(CHEMBL4293688)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University

Curated by ChEMBL
LigandPNGBDBM50466391(CHEMBL4293688)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7RGRPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10651(2-purine deriv. 17 | 4-(6-{[(4-methoxyphenyl)methy...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10650(2-purine deriv. 15 | 5-{6-[(2-methoxyethyl)amino]-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10649(1-(5-{6-[(2-methoxyethyl)amino]-9-(propan-2-yl)-9H...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10648(2-arylpurine deriv. 13 | methyl N-(4-{6-[(2-methox...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10647(2-arylpurine deriv. 12 | N-(2-cyanoethyl)-4-{6-[(2...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10646(2-arylpurine deriv. 11 | 4-{6-[(2-methoxyethyl)ami...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10645(2-arylpurine deriv. 10 | N-(4-{6-[(2-methoxyethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10644(1-(4-{6-[(2-methoxyethyl)amino]-9-(propan-2-yl)-9H...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetGlycogen synthase kinase-3 beta(Rattus norvegicus (rat))
Institut Curie

LigandPNGBDBM10643(2-arylpurine deriv. 8 | 4-{6-[(2-methoxyethyl)amin...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:Kinase activities were assayed in buffers containing substrate, enzyme, and inhibitor at 30 °C in the presence of 15 uM ATP/[gamma-32P] ATP. 32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862DPVPubMed
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50431278(CHEMBL2348264)copy SMILEScopy InChI
Affinity DataKd:  2.90E+3nMAssay Description:Binding affinity to TYRO3 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)copy SMILEScopy InChI
Affinity DataKd:  320nMAssay Description:Binding affinity to nonphosphorylated ABL1 (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50431278(CHEMBL2348264)copy SMILEScopy InChI
Affinity DataKd:  260nMAssay Description:Binding affinity to MER (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Centre Universitaire

Curated by ChEMBL
LigandPNGBDBM50431280(CHEMBL2348263)copy SMILEScopy InChI
Affinity DataKd:  440nMAssay Description:Binding affinity to MET (unknown origin) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V40WJPPubMed
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