Compile Data Set for Download or QSAR
Found 404 with Last Name = 'raab' and Initial = 's'
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50247054(6-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azep...)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Binding affinity to histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50247053(1-(3-(3-(4-chlorophenyl)propoxy)propyl)piperidine ...)copy SMILEScopy InChI
Affinity DataKi:  0.160nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells by [35S]gammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268293((5-(1-cyclobutylpiperidin-4-yloxy)-1-(2,2,2-triflu...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268291((1-(3,4-dichlorophenyl)-5-(1-isopropylpiperidin-4-...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268323((5-(1-cyclopropylpiperidin-4-yloxy)-1-(2,2,2-trifl...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50139391((R)-4-(2-(2-(2-methylpyrrolidin-1-yl)ethyl)benzofu...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Binding affinity to histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Binding affinity to histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268293((5-(1-cyclobutylpiperidin-4-yloxy)-1-(2,2,2-triflu...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269054((4,4-difluoropiperidin-1-yl)(5-(1-isopropylpiperid...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269053((5-(1-isopropylpiperidin-4-yloxy)-1-(2,2,2-trifluo...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268291((1-(3,4-dichlorophenyl)-5-(1-isopropylpiperidin-4-...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327479((S)-7-bromo-2-(cyclopropylmethyl)-8-(1-isopropylpi...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268323((5-(1-cyclopropylpiperidin-4-yloxy)-1-(2,2,2-trifl...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268451(2-(ethoxycarbonyl)-1H-indole-5-carboxylic acid | C...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268947((5-(1-cyclopropylpiperidin-4-yloxy)-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269098((4,4-difluoropiperidin-1-yl)(1-(4-fluorophenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268997((4,4-Difluoropiperidin-1-yl)[5-(1-isopropyl-piperi...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269099(2-(2-(4,4-difluoropiperidine-1-carbonyl)-5-(1-isop...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268815((R)-4'-(3-(3-(dimethylamino)pyrrolidin-1-yl)propox...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding affinity to histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50370569(A-349,821 | A-349821)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding affinity to histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269055((4,4-Difluoropiperidin-1-yl)[1-isopropyl-5-(1-isop...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268996((3,3-difluoropiperidin-1-yl)(5-(1-isopropylpiperid...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268947((5-(1-cyclopropylpiperidin-4-yloxy)-1H-indol-2-yl)...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268997((4,4-Difluoropiperidin-1-yl)[5-(1-isopropyl-piperi...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268996((3,3-difluoropiperidin-1-yl)(5-(1-isopropylpiperid...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269099(2-(2-(4,4-difluoropiperidine-1-carbonyl)-5-(1-isop...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269097((4,4-difluoropiperidin-1-yl)(5-(1-isopropylpiperid...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269053((5-(1-isopropylpiperidin-4-yloxy)-1-(2,2,2-trifluo...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269054((4,4-difluoropiperidin-1-yl)(5-(1-isopropylpiperid...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268948((5-(1-tert-butylpiperidin-4-yloxy)-1H-indol-2-yl)(...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269097((4,4-difluoropiperidin-1-yl)(5-(1-isopropylpiperid...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269098((4,4-difluoropiperidin-1-yl)(1-(4-fluorophenylsulf...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327478((S)-7-bromo-8-(1-isopropylpiperidin-4-yloxy)-4-met...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50240709((R)-4'-(3-(3-(dimethylamino)pyrrolidin-1-yl)propox...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Binding affinity to histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268948((5-(1-tert-butylpiperidin-4-yloxy)-1H-indol-2-yl)(...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327486(8-(1-isopropylpiperidin-4-yloxy)-2-(pyridin-3-ylme...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327473(8-(1-isopropylpiperidin-4-yloxy)-2-(pyridin-4-ylme...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327477((R)-2-(cyclopropylmethyl)-8-(1-isopropylpiperidin-...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268292((1,1-Dioxo-1lambda*6*-thiomorpholin-4-yl)-[5-(1-is...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269096(1-(2-(4,4-difluoropiperidine-1-carbonyl)-5-(1-isop...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50269055((4,4-Difluoropiperidin-1-yl)[1-isopropyl-5-(1-isop...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268949((5-(1-isopropylpiperidin-4-yloxy)-1H-indol-2-yl)(m...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268452((4-cyclobutylpiperazin-1-yl)(2-(morpholine-4-carbo...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327475((S)-8-(1-isopropylpiperidin-4-yloxy)-3-methyl-3,4-...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327487(2-(2-fluorobenzyl)-8-(1-isopropylpiperidin-4-yloxy...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50327488(8-(1-isopropylpiperidin-4-yloxy)-2-(pyridin-2-ylme...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-RAMH from human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571C7NPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268950(CHEMBL522715 | azepan-1-yl(5-(1-isopropylpiperidin...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268451(2-(ethoxycarbonyl)-1H-indole-5-carboxylic acid | C...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268998((1,1-Dioxo-1lambda*6*-thiomorpholin-4-yl)-[5-(1-is...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche Ltd.

Curated by ChEMBL
LigandPNGBDBM50268949((5-(1-isopropylpiperidin-4-yloxy)-1H-indol-2-yl)(m...)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from rat recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB46NQPubMed
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