Compile Data Set for Download or QSAR
Found 29 with Last Name = 'saul' and Initial = 's'
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562897(CHEMBL4740761)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562898(CHEMBL4778276)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562894(CHEMBL4762694)copy SMILES
Affinity DataIC50: 3.80nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562893(CHEMBL4764705)copy SMILES
Affinity DataIC50: 7.70nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562895(CHEMBL4794323)copy SMILES
Affinity DataIC50: 8.80nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562914(CHEMBL4745919)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562913(CHEMBL4745028)copy SMILES
Affinity DataIC50: 13nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562905(CHEMBL4800032)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562896(CHEMBL4779229)copy SMILES
Affinity DataIC50: 17nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562907(CHEMBL4752286)copy SMILES
Affinity DataIC50: 35nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562908(CHEMBL4784439)copy SMILES
Affinity DataIC50: 37nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562906(CHEMBL4755134)copy SMILES
Affinity DataIC50: 39nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50524284(CHEMBL4443342)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of NanoBRET tracer 5 binding to NL-fused GAK (unknown origin) expressed in HEK293 cells measured after 2 hrs by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50086268(CHEMBL3425867)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562911(CHEMBL4790097)copy SMILES
Affinity DataIC50: 62nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562904(CHEMBL4760106)copy SMILES
Affinity DataIC50: 69nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562901(CHEMBL4782363)copy SMILES
Affinity DataIC50: 74nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562910(CHEMBL4753946)copy SMILES
Affinity DataIC50: 78nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562915(CHEMBL4756485)copy SMILES
Affinity DataIC50: 78nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562909(CHEMBL4799769)copy SMILES
Affinity DataIC50: 85nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562902(CHEMBL4777592)copy SMILES
Affinity DataIC50: 190nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562912(CHEMBL4747444)copy SMILES
Affinity DataIC50: 360nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562917(CHEMBL4800155)copy SMILES
Affinity DataIC50: 500nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562900(CHEMBL4798132)copy SMILES
Affinity DataIC50: 900nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562899(CHEMBL4782593)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562916(CHEMBL4745993)copy SMILES
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562903(CHEMBL4759566)copy SMILES
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataKd:  3.10nMAssay Description:Binding affinity to GAK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed