Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 0.0210nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 2.14nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 3.36nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 4.13nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 5.13nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 7.12nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 27.1nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 30.3nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 49.5nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 118nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 382nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 384nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to Serotonin 5-HT1A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 423nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 547nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 670nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 733nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 2.60E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 3.51E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 3.90E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 4.01E+3nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Affinity DataKi: 4.51E+3nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-spiperone binding to Dopamine D2 receptor from rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 0.4 nM [3H]-ketanserin binding to Serotonin 5-HT2A receptor from rat brain cortexMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: 1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to Dopamine D1 receptor from rat striatumMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Università di Napoli "Federico II"
Curated by ChEMBL
Università di Napoli "Federico II"
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 1 nM [3H]-mesulergine binding to Serotonin 5-HT2C receptor from rat brain cortexMore data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Mashhad University of Medical Sciences
Curated by ChEMBL
Mashhad University of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using BML-KI104 Fluor de Lys as substrate by fluorescence-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of full length HDAC3 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Inhibition of full length HDAC1 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Antagonist potency against carbachol induced inhibition of electrically stimulated guinea pig atria Muscarinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 179nMAssay Description:Inhibition of full length HDAC2 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of mPGES1 in IL-1beta-stimulated human A549 cell microsomes using PGH2 as substrate assessed as reduction in PGE2 production preincubated ...More data for this Ligand-Target Pair