Affinity DataIC50: 1nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Mahidol University
Curated by ChEMBL
Mahidol University
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human HMGR catalytic domain using 800 uM HMG-CoA as substrate measured every 20 secs for 10 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Prince of Songkla University
Curated by ChEMBL
Prince of Songkla University
Curated by ChEMBL
Affinity DataIC50: 5.86E+4nMAssay Description:Inhibition of CFTR-mediated forskolin-induced chloride secretion in human T84 cells after 15 mins by short-circuit current analysisMore data for this Ligand-Target Pair
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Homo sapiens (Human))
Mahidol University
Curated by ChEMBL
Mahidol University
Curated by ChEMBL
Affinity DataIC50: 3.87E+5nMAssay Description:Inhibition of human HMGR catalytic domain using 800 uM HMG-CoA as substrate measured every 20 secs for 10 minsMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 530nMAssay Description:Inhibition of 8Fluo-cAMP binding to recombinant human His-tagged EPAC1 (157 to 881 residues) expressed in Escherichia coli measured after 5 mins by f...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 3.87E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 5.62E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to recombinant human His-tagged EPAC1 (157 to 881 residues) expressed in Escherichia coli measured after 5 mins by f...More data for this Ligand-Target Pair
TargetPotassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Activation of recombinant mouse HCN2 expressed in Xenopus laevis oocyte assessed as increase in current amplitude at -30 mV holding potential by patc...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 2.36E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 6.40E+3nMAssay Description:Activation of recombinant rat CNGA2 expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch-clamp electrophysiology met...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Activation of recombinant rat CNGA2/CNGA4/CNGB1b heterotetramer expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 2.54E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to recombinant human His-tagged EPAC1 (157 to 881 residues) expressed in Escherichia coli measured after 5 mins by f...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 540nMAssay Description:Activation of recombinant rat CNGA2 expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch-clamp electrophysiology met...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 630nMAssay Description:Activation of recombinant rat CNGA2/CNGA4/CNGB1b heterotetramer expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 780nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 2.75E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to recombinant human His-tagged EPAC1 (157 to 881 residues) expressed in Escherichia coli measured after 5 mins by f...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 4.98E+3nMAssay Description:Activation of recombinant rat CNGA2/CNGA4/CNGB1b heterotetramer expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Activation of recombinant rat CNGA2/CNGA4/CNGB1b heterotetramer expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Activation of recombinant rat CNGA2/CNGA4/CNGB1b heterotetramer expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 5.31E+4nMAssay Description:Activation of recombinant rat CNGA2 expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch-clamp electrophysiology met...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 1.54E+4nMAssay Description:Activation of recombinant rat CNGA2 expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch-clamp electrophysiology met...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 2.06E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 2.08E+3nMAssay Description:Activation of recombinant rat CNGA2 expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch-clamp electrophysiology met...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 1.09E+3nMAssay Description:Inhibition of 8Fluo-cAMP binding to recombinant human His-tagged EPAC1 (157 to 881 residues) expressed in Escherichia coli measured after 5 mins by f...More data for this Ligand-Target Pair
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