TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Reversible mixed-type inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 ...More data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Competitive inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 mins...More data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.610nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.720nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.760nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.34nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 2.64nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2B8594WPubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
The First Affiliated Hospital of Guangzhou Medical University
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 minsMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)