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Found 191 with Last Name = 'zeng' and Initial = 's'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283545(CHEMBL4162340)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Reversible mixed-type inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50335784(2-[6-(3-Aminopiperidin-1-yl)-3-methyl-2,4-dioxo-3,...)copy SMILEScopy InChI
Affinity DataKi:  5.10nMAssay Description:Competitive inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 mins...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))TBA
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)copy SMILEScopy InChI
Affinity DataKi:  42nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))TBA
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))TBA
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)copy SMILEScopy InChI
Affinity DataIC50: 0.370nMMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))TBA
LigandPNGBDBM50590371(CHEMBL5182618)copy SMILES
Affinity DataIC50: 0.540nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283680(CHEMBL4164470)copy SMILEScopy InChI
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283674(CHEMBL4176578)copy SMILEScopy InChI
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283666(CHEMBL4169845)copy SMILEScopy InChI
Affinity DataIC50: 0.610nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283675(CHEMBL4175111)copy SMILEScopy InChI
Affinity DataIC50: 0.720nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283673(CHEMBL4165967)copy SMILEScopy InChI
Affinity DataIC50: 0.760nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283543(CHEMBL4172793)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283678(CHEMBL4162971)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283671(CHEMBL4169403)copy SMILEScopy InChI
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))TBA
LigandPNGBDBM185674(4-[4-[(5-tert-butyl-2-quinolin-6-ylpyrazol-3-yl)ca...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
LigandPNGBDBM50590370(K-0706 | K0706 | Sco-088 | VODOBATINIB | Vodobatin...)copy SMILES
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283672(CHEMBL4164893)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50381853(CHEMBL2023067)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50335784(2-[6-(3-Aminopiperidin-1-yl)-3-methyl-2,4-dioxo-3,...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283677(CHEMBL4173673)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283544(CHEMBL4173272)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283630(CHEMBL4161924)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50431782(CHEMBL2347039)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78GMRPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283664(CHEMBL4161474)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283676(CHEMBL4165359)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283545(CHEMBL4162340)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50381855(CHEMBL2023066)copy SMILEScopy InChI
Affinity DataIC50: 2.34nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283668(CHEMBL4169618)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19D0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50381854(CHEMBL2022467)copy SMILEScopy InChI
Affinity DataIC50: 2.64nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B8594WPubMed
TargetAurora kinase A(Homo sapiens (Human))TBA
LigandPNGBDBM209859(4-N-(5-cyclopropyl-1H-pyrazol-3-yl)-6-(4-methylpip...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human DPP4 after 10 minsMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))TBA
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))TBA
LigandPNGBDBM50355496(CHEMBL1908397)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))TBA
LigandPNGBDBM50243388(AT-9283 | US10981896, Compound AT9283)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50431785(CHEMBL2347036)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78GMRPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))TBA
LigandPNGBDBM185674(4-[4-[(5-tert-butyl-2-quinolin-6-ylpyrazol-3-yl)ca...)copy SMILEScopy InChI
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))TBA
LigandPNGBDBM209859(4-N-(5-cyclopropyl-1H-pyrazol-3-yl)-6-(4-methylpip...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))TBA
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89HCMPubMedDrugBank
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