Compile Data Set for Download or QSAR
Found 96 with Last Name = 'hwang' and Initial = 'sb'
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))copy SMILEScopy InChI
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))copy SMILEScopy InChI
Affinity DataKi:  5.48nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  12.2nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  14.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)copy SMILEScopy InChI
Affinity DataKi:  79.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  152nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  205nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  1.11E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021572((2S,3S)-2-(3,4-Dimethoxy-phenyl)-3-methyl-5-propyl...)copy SMILEScopy InChI
Affinity DataIC50: 0nMAssay Description:Inhibitor concentration required to block 50% of the specific [3H]PAF binding to rabbit platelet membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25T3M2XPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408421(CHEMBL2113725)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286666(CHEMBL347382 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:In vitro inhibition of 5-lipoxygenase in RBL-2H3 (Rat basophilic leukaemia) cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286666(CHEMBL347382 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408414(CHEMBL2113720)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286665(CHEMBL160692 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286665(CHEMBL160692 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of 5-lipoxygenase in RBL-2H3 (Rat basophilic leukaemia) cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286669(5-lipoxygenase inhibitor | CHEMBL348609)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50408417(CHEMBL2113724)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50408419(CHEMBL2113723)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408413(CHEMBL2113727)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50002831((2R,5R)-2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of PAF receptor binding to rabbit platelet plasma membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X63KZSPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408419(CHEMBL2113723)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408418(CHEMBL2113722)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408422(CHEMBL2113721)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408424(CHEMBL2113733)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286661(CHEMBL160290 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286661(CHEMBL160290 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286667(CHEMBL155851 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286667(CHEMBL155851 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286668(CHEMBL160218 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286668(CHEMBL160218 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50408422(CHEMBL2113721)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:In vitro inhibition of 5-lipoxygenase in RBL-2H3 (Rat basophilic leukaemia) cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408423(CHEMBL2113726)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408415(CHEMBL2113730)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50408418(CHEMBL2113722)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408417(CHEMBL2113724)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286658(5-lipoxygenase inhibitor | CHEMBL155760)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50408413(CHEMBL2113727)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:5-lipoxygenase inhibitory activity determined by measuring the conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cell using thin-layer ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286660(5-lipoxygenase inhibitor | CHEMBL160839)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286659(5-lipoxygenase inhibitor | CHEMBL434090)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50405462(CHEMBL2115332)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibitor concentration required to block 50 of the specific [3H]PAF binding to rabbit platelet membranes.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25T3M2XPubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50408415(CHEMBL2113730)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286656(5-lipoxygenase inhibitor | CHEMBL160571)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23778QB
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)copy SMILEScopy InChI
Affinity DataIC50: 94nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50408414(CHEMBL2113720)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6JH2PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50001747((+)-Kadsurenone | (Kadsurenone)5-Allyl-2-(3,4-dime...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibitor concentration required to block 50% of the specific [3H]PAF binding, obtained as natural product.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q25T3M2XPubMed
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