Compile Data Set for Download or QSAR
Found 680 with Last Name = 'cheon' and Initial = 'sh'
TargetD(3) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50111766(CHEMBL3605331)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D3 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F1XPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50111767(CHEMBL3605344)copy SMILEScopy InChI
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D3 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F1XPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50111765(CHEMBL3605327)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D3 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F1XPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50111766(CHEMBL3605331)copy SMILEScopy InChI
Affinity DataKi:  175nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D2 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F1XPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50111767(CHEMBL3605344)copy SMILEScopy InChI
Affinity DataKi:  197nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D2 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F1XPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500112(CHEMBL3739820)copy SMILEScopy InChI
Affinity DataKi:  270nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D3 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500110(CHEMBL3740498)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D3 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50131925(1H-Indole-2-carboxylic acid {4-[4-(2,4-dichloro-ph...)copy SMILEScopy InChI
Affinity DataKi:  410nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D3 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500111(CHEMBL3740360)copy SMILEScopy InChI
Affinity DataKi:  810nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D3 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500110(CHEMBL3740498)copy SMILEScopy InChI
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D2 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50111765(CHEMBL3605327)copy SMILEScopy InChI
Affinity DataKi:  5.59E+3nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D2 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F1XPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500111(CHEMBL3740360)copy SMILEScopy InChI
Affinity DataKi:  6.23E+3nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D2 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50131925(1H-Indole-2-carboxylic acid {4-[4-(2,4-dichloro-ph...)copy SMILEScopy InChI
Affinity DataKi: >2.39E+4nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D2 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500112(CHEMBL3739820)copy SMILEScopy InChI
Affinity DataKi:  7.96E+4nMAssay Description:Displacement of [3H]-sulpiride from human dopamine D2 receptor expressed in HEK293 cells after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J38WK1PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50041917(4-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:In vitro PAF antagonistic activity by determining [3H]-PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27P8XFQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMedDrugBank
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048175(CHEMBL3310482)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048172(CHEMBL3310485)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048178(CHEMBL3310489)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048171(CHEMBL3310484)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM22417(3-(2-methoxyphenoxy)-N-methyl-3-phenylpropan-1-ami...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048178(CHEMBL3310489)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048169(CHEMBL3310483)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048176(CHEMBL3310487)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048175(CHEMBL3310482)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of DA reuptake at human DAT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048174(CHEMBL3310486)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048179(CHEMBL3310490)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048168(CHEMBL3310478)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048135(CHEMBL3309701)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048172(CHEMBL3310485)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of DA reuptake at human DAT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMedDrugBank
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048136(CHEMBL3309702)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of norepinephrine reuptake at human NET expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048172(CHEMBL3310485)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048176(CHEMBL3310487)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048177(CHEMBL3310488)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048179(CHEMBL3310490)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of re-uptake of [3H]-DA at human DAT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50041919(6-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-3...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:In vitro PAF antagonistic activity by determining [3H]-PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27P8XFQPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of [3H]-5-dopamine reuptake in human DAT expressed in HEK293 cells by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN47BSPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048171(CHEMBL3310484)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048169(CHEMBL3310483)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50041924(7-Methyl-4-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:In vitro PAF antagonistic activity by determining [3H]-PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27P8XFQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048175(CHEMBL3310482)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048136(CHEMBL3309702)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of DA reuptake at human DAT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048135(CHEMBL3309701)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of DA reuptake at human DAT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50117973(CHEMBL3612829)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50117973(CHEMBL3612829)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction of serotonin reuptake using [3H]-SERT after 15 mins by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78H1JPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50048174(CHEMBL3310486)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Inhibition of serotonin reuptake at human SERT expressed in HEK293 cells after 15 mins by fluorescence neurotransmitter transporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1MHHPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50041916(2,2-Dimethyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:In vitro PAF antagonistic activity by determining [3H]-PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27P8XFQPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Sandoz Research Institute

Curated by ChEMBL
LigandPNGBDBM50041921(5-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:In vitro PAF antagonistic activity by determining [3H]-PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27P8XFQPubMed
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