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Found 103 with Last Name = 'verhelst' and Initial = 'sh'
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50514789(CHEMBL4564966)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:Inhibition of full length wild type human N-terminal GST-tagged MALT1 catalytic domain (325 to 760 residues) expressed in Escherichia coli BL21 (DE3)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0DBRPubMed
TargetCathepsin B(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50514790(CHEMBL4565998)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of recombinant human cathepsin B expressed in Escherichia coli BL21 (DE3) using zRR-AMC as substrate measured after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0DBRPubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50514790(CHEMBL4565998)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of full length wild type human N-terminal GST-tagged MALT1 catalytic domain (325 to 760 residues) expressed in Escherichia coli BL21 (DE3)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0DBRPubMed
TargetMucosa-associated lymphoid tissue lymphoma translocation protein 1(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50514791(CHEMBL3814336)copy SMILEScopy InChI
Affinity DataKi:  340nMAssay Description:Inhibition of full length wild type human N-terminal GST-tagged MALT1 catalytic domain (325 to 760 residues) expressed in Escherichia coli BL21 (DE3)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0DBRPubMed
TargetCathepsin B(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50514791(CHEMBL3814336)copy SMILEScopy InChI
Affinity DataKi:  630nMAssay Description:Inhibition of recombinant human cathepsin B expressed in Escherichia coli BL21 (DE3) using zRR-AMC as substrate measured after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0DBRPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50544647(CHEMBL4634122)copy SMILEScopy InChI
Affinity DataKi:  2.96E+3nMAssay Description:Inhibition of human neutrophil elastase using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P357NPubMed
TargetCathepsin B(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50514789(CHEMBL4564966)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of recombinant human cathepsin B expressed in Escherichia coli BL21 (DE3) using zRR-AMC as substrate measured after 2 hrs by fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0DBRPubMed
TargetMyeloblastin(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50544646(CHEMBL4635621)copy SMILEScopy InChI
Affinity DataKi:  2.65E+4nMAssay Description:Inhibition of human proteinase 3 using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P357NPubMed
TargetNeutrophil elastase(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50544646(CHEMBL4635621)copy SMILEScopy InChI
Affinity DataKi:  5.10E+4nMAssay Description:Inhibition of human neutrophil elastase using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P357NPubMed
TargetMyeloblastin(Homo sapiens (Human))
KU Leuven

Curated by ChEMBL
LigandPNGBDBM50544648(CHEMBL4636971)copy SMILEScopy InChI
Affinity DataKi:  8.38E+4nMAssay Description:Inhibition of human proteinase 3 using flurogenic substrate as elastase substrate V by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P357NPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591345(CHEMBL5196519)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591344(CHEMBL5208857)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591341(CHEMBL5177372)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591337(CHEMBL5192445)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591336(CHEMBL5179027)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591331(CHEMBL5197282)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591344(CHEMBL5208857)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591341(CHEMBL5177372)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591340(CHEMBL5203787)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591337(CHEMBL5192445)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591336(CHEMBL5179027)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591334(CHEMBL5191146)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591331(CHEMBL5197282)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591330(CHEMBL5197431)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591327(CHEMBL5177544)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM158481(US9029401, 1728 (t-TUCB))copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM409005(US10377744, Compound No. 26 | US11123311, Compound...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50217448(CHEMBL242459 | US9029401, 1471 (t-AUCB) | trans-4-...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591345(CHEMBL5196519)copy SMILES
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591340(CHEMBL5203787)copy SMILES
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591335(CHEMBL5179500)copy SMILES
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591333(CHEMBL5197313)copy SMILES
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591338(CHEMBL5203245)copy SMILES
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591338(CHEMBL5203245)copy SMILES
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591332(CHEMBL5195267)copy SMILES
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591334(CHEMBL5191146)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591333(CHEMBL5197313)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591343(CHEMBL5209279)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591328(CHEMBL5193653)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591329(CHEMBL5179393)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591335(CHEMBL5179500)copy SMILES
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591332(CHEMBL5195267)copy SMILES
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591329(CHEMBL5179393)copy SMILES
Affinity DataIC50: 2.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50581722(CHEMBL5081815)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50581722(CHEMBL5081815)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591330(CHEMBL5197431)copy SMILES
Affinity DataIC50: 6.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50191854(CHEMBL436774 | N-(1-acetyl-piperidin-4-yl)-N'-(ada...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50591339(CHEMBL5169759)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))TBA
LigandPNGBDBM50591328(CHEMBL5193653)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VHVPubMed
TargetAcyl-protein thioesterase 2(Mus musculus)TBA
LigandPNGBDBM50547464(CHEMBL4776695)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of FP-Rh binding to APT-1/2 in mouse brain cytosolic fraction preincubated for 1 hr followed by FP-Rh addition and measured after 1 hr by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8C8BPubMed
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