Compile Data Set for Download or QSAR
Found 132 with Last Name = 'shaw' and Initial = 'sj'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251456(CHEMBL4084955)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251453(CHEMBL4079572)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251457(CHEMBL4105629)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251509(CHEMBL4064316)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Kosan Biosciences, Inc.

Curated by ChEMBL
LigandPNGBDBM50299505(3 9-dihydro-N-desmethyl-N-isopropylerythromycin A ...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human ERG expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C1XT1PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251436(CHEMBL4091320)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251451(CHEMBL4069163)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetFlap endonuclease 1 [1-336](Homo sapiens (Human))
University of Sheffield

LigandPNGBDBM197162(3-hydroxy-1-(4-methoxybenzyl)quinazoline-2,4(1H,3H...)copy SMILEScopy InChI
Affinity DataIC50: 16.9nMpH: 7.5Assay Description:Reaction mixtures containing twelve different concentrations of FAM-labeled DF1 (Supplementary Fig. 5a) substrate were prepared in reaction buffer (R...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4H88PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50081190(CHEMBL3421979)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetFlap endonuclease 1 [1-336](Homo sapiens (Human))
University of Sheffield

LigandPNGBDBM197161(1-(cyclopropylmethyl)-3-hydroxyquinazoline-2,4(1H,...)copy SMILEScopy InChI
Affinity DataIC50: 30nMpH: 7.5Assay Description:Reaction mixtures containing twelve different concentrations of FAM-labeled DF1 (Supplementary Fig. 5a) substrate were prepared in reaction buffer (R...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4H88PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Kosan Biosciences, Inc.

Curated by ChEMBL
LigandPNGBDBM50344942(CHEMBL532 | E-MYCIN E | ERYTHROMYCIN | ERYTHROMYCI...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of human ERG expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C1XT1PubMedDrugBank
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251479(CHEMBL4073997)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetFlap endonuclease 1 [1-336](Homo sapiens (Human))
University of Sheffield

LigandPNGBDBM50157840(1-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-3-...)copy SMILEScopy InChI
Affinity DataIC50: 46.4nMpH: 7.5Assay Description:Reaction mixtures containing twelve different concentrations of FAM-labeled DF1 (Supplementary Fig. 5a) substrate were prepared in reaction buffer (R...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251477(CHEMBL4075648)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251458(CHEMBL4087456)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251504(CHEMBL4098505)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251485(CHEMBL4080488)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50347796(CHEMBL1802963)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251452(CHEMBL4077010)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251480(CHEMBL4086818)copy SMILEScopy InChI
Affinity DataIC50: 94nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251476(CHEMBL4095674)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251478(CHEMBL4072138)copy SMILEScopy InChI
Affinity DataIC50: 138nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251475(CHEMBL4090889)copy SMILEScopy InChI
Affinity DataIC50: 242nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251486(CHEMBL4066607)copy SMILEScopy InChI
Affinity DataIC50: 277nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251507(CHEMBL4094549)copy SMILEScopy InChI
Affinity DataIC50: 285nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251510(CHEMBL4095156)copy SMILEScopy InChI
Affinity DataIC50: 351nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251508(CHEMBL4065388)copy SMILEScopy InChI
Affinity DataIC50: 406nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Kosan Biosciences, Inc.

Curated by ChEMBL
LigandPNGBDBM50299517(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 411nMAssay Description:Inhibition of human ERG expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C1XT1PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251506(CHEMBL4095479)copy SMILEScopy InChI
Affinity DataIC50: 443nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM10844(4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)copy SMILEScopy InChI
Affinity DataIC50: 588nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251509(CHEMBL4064316)copy SMILEScopy InChI
Affinity DataIC50: 660nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251503(CHEMBL4066075)copy SMILEScopy InChI
Affinity DataIC50: 790nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251451(CHEMBL4069163)copy SMILEScopy InChI
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251457(CHEMBL4105629)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM327994(N-(1-(4- cyanobenzyl)piperidin-4- yl)-5-(4-(4- met...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1HM7PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251484(CHEMBL4074685)copy SMILEScopy InChI
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251505(CHEMBL4068096)copy SMILEScopy InChI
Affinity DataIC50: 2.14E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251482(CHEMBL4098364)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251481(CHEMBL4069088)copy SMILEScopy InChI
Affinity DataIC50: 2.94E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251436(CHEMBL4091320)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))TBA
LigandPNGBDBM327998(N-(1-(4- cyanobenzyl)piperidin-4- yl)-5-(4-(4- cya...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1HM7PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251502(CHEMBL4103831)copy SMILEScopy InChI
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251452(CHEMBL4077010)copy SMILEScopy InChI
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251478(CHEMBL4072138)copy SMILEScopy InChI
Affinity DataIC50: 5.16E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251476(CHEMBL4095674)copy SMILEScopy InChI
Affinity DataIC50: 7.58E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251483(CHEMBL4102903)copy SMILEScopy InChI
Affinity DataIC50: 7.96E+3nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251506(CHEMBL4095479)copy SMILEScopy InChI
Affinity DataIC50: 7.96E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251456(CHEMBL4084955)copy SMILEScopy InChI
Affinity DataIC50: 9.23E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50251477(CHEMBL4075648)copy SMILEScopy InChI
Affinity DataIC50: 9.61E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0CFPPubMed
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