Compile Data Set for Download or QSAR
Found 21 with Last Name = 'nahorski' and Initial = 'sr'
LigandPNGBDBM50132166(1,2,4,5-InsP4 | CHEMBL100498 | Phosphoric acid mon...)copy SMILEScopy InChI
Affinity DataKi:  26.4nMAssay Description:Compound was evaluated for its ability to displace [3H]Ins(1,4,5)P3 from membranes prepared from bovine adrenal corticlesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M08F4
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50407003(CHEMBL2092837)copy SMILEScopy InChI
Affinity DataKi:  3.90E+3nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50046068(1D-3-deoxy- 1D-myo-Inositol 1,4,5-trisphosphate)copy SMILEScopy InChI
Affinity DataKi:  1.15E+4nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (S substrate)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50075183(1,4,5-Insp3 | 1D-myo-inositol 1,4,5-triphosphate |...)copy SMILEScopy InChI
Affinity DataKi:  1.50E+4nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (S substrate)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50046075(1D-2,3,6--trioxy- 1D-myo-Inositol 1,4,5-trisphosph...)copy SMILEScopy InChI
Affinity DataKi:  1.65E+4nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (S substrate)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50046074(1D-2,3,6--trideoxy- 1D-myo-Inositol 1,4,5-trisphos...)copy SMILEScopy InChI
Affinity DataKi:  8.14E+4nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (S substrate)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50046070((1R,2R,4R)-Cyclohexane-1,2,4-tris (methlyenephosph...)copy SMILEScopy InChI
Affinity DataKi:  1.44E+5nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (R metabolically resistant)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50046073(Benzene-1,2,4-tris (methylenephosphonate))copy SMILEScopy InChI
Affinity DataKi:  1.48E+5nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (R metabolically resistant)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50046072((1R,2R,4R)-Cyclohexane-1,2,4-tris (methylenephosph...)copy SMILEScopy InChI
Affinity DataKi:  5.35E+5nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (R metabolically resistant)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol-trisphosphate 3-kinase C(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50040911((+)-myo-inositol 1,4,5-trisphosphorothioate | (-)-...)copy SMILEScopy InChI
Affinity DataKi:  9.78E+5nMAssay Description:Tested for the ability to inhibit Ins(1,4,5)P 3-phosphataseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8849
TargetInositol polyphosphate-5-phosphatase A(Homo sapiens (Human))
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50407004(CHEMBL2092922)copy SMILEScopy InChI
Affinity DataKi: >1.00E+8nMAssay Description:Tested for inhibition of 5-phosphatase isolated from human erythrocyte membrane (R metabolically resistant)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2T72J2RPubMed
TargetInositol 1,4,5-trisphosphate receptor type 2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50075183(1,4,5-Insp3 | 1D-myo-inositol 1,4,5-triphosphate |...)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:The compound was tested for inhibitory activity against IInositol 1,4,5-trisphosphate receptor in SH-SY5Y cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V5MPubMed
TargetInositol 1,4,5-trisphosphate receptor type 2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50221652(CHEMBL3349691)copy SMILEScopy InChI
Affinity DataIC50: 26.5nMAssay Description:The compound was tested for inhibitory activity against Inositol 1,4,5-trisphosphate receptor in SH-SY5Y cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V5MPubMed
TargetInositol 1,4,5-trisphosphate receptor type 2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50221652(CHEMBL3349691)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:The compound was tested for inhibitory activity against Inositol 1,4,5-trisphosphate receptor in SH-SY5Y cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V5MPubMed
TargetInositol 1,4,5-trisphosphate receptor type 2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50075183(1,4,5-Insp3 | 1D-myo-inositol 1,4,5-triphosphate |...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:The compound was tested for inhibitory activity against Inositol 1,4,5-trisphosphate receptor in L15 cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V5MPubMed
TargetInositol 1,4,5-trisphosphate receptor type 2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50075183(1,4,5-Insp3 | 1D-myo-inositol 1,4,5-triphosphate |...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:The compound was tested for inhibitory activity against Inositol 1,4,5-trisphosphate receptor in SH-SY5Y cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V5MPubMed
TargetType 1 InsP3 receptor isoform S2(Sus scrofa)
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50040911((+)-myo-inositol 1,4,5-trisphosphorothioate | (-)-...)copy SMILEScopy InChI
Affinity DataIC50: 61nMpH: 7.6Assay Description:Binding affinity against IP3 receptor in pig cerebellar membranes at a pH of 7.6 using [3H]Ins(1,4,5)P3 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PN3PubMed
TargetType 1 InsP3 receptor isoform S2(Sus scrofa)
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50040911((+)-myo-inositol 1,4,5-trisphosphorothioate | (-)-...)copy SMILEScopy InChI
Affinity DataIC50: 78nMpH: 6.8Assay Description:Binding affinity against IP3 receptor in pig cerebellar membranes at a pH of 6.8 using [3H]Ins(1,4,5)P3 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PN3PubMed
TargetInositol 1,4,5-trisphosphate receptor type 2(Homo sapiens (Human))
University of Bath

Curated by ChEMBL
LigandPNGBDBM50472223(CHEMBL1160286)copy SMILEScopy InChI
Affinity DataIC50: 172nMAssay Description:The compound was tested for inhibitory activity against Inositol 1,4,5-trisphosphate receptor in L15 cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V5MPubMed
TargetType 1 InsP3 receptor isoform S2(Sus scrofa)
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50040909(D-3-amino-3-deoxy-myo-inositol 1,4,5-trisphosphoro...)copy SMILEScopy InChI
Affinity DataIC50: 5.65E+3nMpH: 7.6Assay Description:Binding affinity against IP3 receptor in pig cerebellar membranes at a pH of 7.6 using [3H]Ins(1,4,5)P3 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PN3PubMed
TargetType 1 InsP3 receptor isoform S2(Sus scrofa)
Mayo Foundation for Medical Education and Research

Curated by ChEMBL
LigandPNGBDBM50040909(D-3-amino-3-deoxy-myo-inositol 1,4,5-trisphosphoro...)copy SMILEScopy InChI
Affinity DataIC50: 9.11E+3nMpH: 6.8Assay Description:Binding affinity against IP3 receptor in pig cerebellar membranes at a pH of 6.8 using [3H]Ins(1,4,5)P3 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PN3PubMed