Compile Data Set for Download or QSAR
Found 91 with Last Name = 'le quement' and Initial = 'st'
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498101(CHEMBL3403862)copy SMILEScopy InChI
Affinity DataIC50: 3.81E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498105(CHEMBL3403858)copy SMILEScopy InChI
Affinity DataIC50: 4.25E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498098(CHEMBL3403859)copy SMILEScopy InChI
Affinity DataIC50: 4.99E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498104(CHEMBL3403865)copy SMILEScopy InChI
Affinity DataIC50: 5.82E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498097(CHEMBL3403860)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498102(CHEMBL3403856)copy SMILEScopy InChI
Affinity DataIC50: 6.78E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498100(CHEMBL3403864)copy SMILEScopy InChI
Affinity DataIC50: 6.92E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498103(CHEMBL3403861)copy SMILEScopy InChI
Affinity DataIC50: 8.89E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498099(CHEMBL3403868)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+6nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)copy SMILEScopy InChI
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)copy SMILEScopy InChI
Affinity DataEC50:  24nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250212(CHEMBL4089119)copy SMILEScopy InChI
Affinity DataEC50:  185nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250213(CHEMBL4104927)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250211(CHEMBL4100221)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)copy SMILEScopy InChI
Affinity DataEC50:  35nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250205(CHEMBL4067491)copy SMILEScopy InChI
Affinity DataEC50:  110nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250206(CHEMBL4060816)copy SMILEScopy InChI
Affinity DataEC50:  9.20nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250207(CHEMBL4082585)copy SMILEScopy InChI
Affinity DataEC50:  64nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250208(CHEMBL4062443)copy SMILEScopy InChI
Affinity DataEC50:  792nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250209(CHEMBL4090425)copy SMILEScopy InChI
Affinity DataEC50:  124nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250210(CHEMBL4087072)copy SMILEScopy InChI
Affinity DataEC50:  730nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250182(CHEMBL4077331)copy SMILEScopy InChI
Affinity DataEC50:  685nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)copy SMILEScopy InChI
Affinity DataEC50:  29nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)copy SMILEScopy InChI
Affinity DataEC50:  633nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250199(CHEMBL4092477)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250182(CHEMBL4077331)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250210(CHEMBL4087072)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250201(CHEMBL4070639)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250182(CHEMBL4077331)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250199(CHEMBL4092477)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)copy SMILEScopy InChI
Affinity DataEC50:  375nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250201(CHEMBL4070639)copy SMILEScopy InChI
Affinity DataEC50:  137nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250202(CHEMBL4074680)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250203(CHEMBL4083755)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250204(CHEMBL4060937)copy SMILEScopy InChI
Affinity DataEC50:  916nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250213(CHEMBL4104927)copy SMILEScopy InChI
Affinity DataEC50:  291nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250208(CHEMBL4062443)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250207(CHEMBL4082585)copy SMILEScopy InChI
Affinity DataEC50:  821nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250202(CHEMBL4074680)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250203(CHEMBL4083755)copy SMILEScopy InChI
Affinity DataEC50:  89nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250212(CHEMBL4089119)copy SMILEScopy InChI
Affinity DataEC50:  720nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)copy SMILEScopy InChI
Affinity DataEC50:  162nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)copy SMILEScopy InChI
Affinity DataEC50:  635nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250207(CHEMBL4082585)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250208(CHEMBL4062443)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataEC50:  34nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250204(CHEMBL4060937)copy SMILEScopy InChI
Affinity DataEC50:  160nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
Displayed 1 to 50 (of 91 total ) | Next | Last >>
Jump to: