TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 0.290nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 0.390nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human JAK1 using poly[Glu:Tyr] (4:1) as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 0.740nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human JAK2 using poly[Glu:Tyr] (4:1) as substrate in presence of 10 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Eberhard Karls University T£bingen
Curated by ChEMBL
Eberhard Karls University T£bingen
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate in presence of 200 uM [gamma33P]ATP by radiometric methodMore data for this Ligand-Target Pair
In DepthDetails
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