Compile Data Set for Download or QSAR
Found 88 with Last Name = 'hoshino' and Initial = 't'
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Chiba University

Curated by ChEMBL
LigandPNGBDBM105203(6-(4-Fluorophenyl)-3-hydroxy-5-[4-(1H-1, 2, 3, 4-t...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of Influenza A/Puerto Rico/8/34 (H1N1) PA N-terminal domain endonuclease activity expressed in Escherichia coli BL21 (RIL) cells using (6-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87CK3PubMed
TargetHistone deacetylase 1(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)copy SMILEScopy InChI
Affinity DataIC50: 36.6nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetHistone deacetylase 4(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)copy SMILEScopy InChI
Affinity DataIC50: 62.9nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetHistone deacetylase 6(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM19130((2E,4E,6R)-7-[4-(dimethylamino)phenyl]-N-hydroxy-4...)copy SMILEScopy InChI
Affinity DataIC50: 83.3nMAssay Description:Inhibition of human HDAC6 expressed in 293T cellsMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482161(CHEMBL1082256)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated ribonuclease H activity by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482160(CHEMBL1082257)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of HIV1 reverse transcriptase-associated ribonuclease H activity by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482159(CHEMBL1082255)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482159(CHEMBL1082255)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483220(CHEMBL1535664)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetHistone deacetylase 1(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50377384(AZUMAMIDE C)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetHistone deacetylase 1(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50372469(AZUMAMIDE E)copy SMILEScopy InChI
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetHistone deacetylase 1(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50377383(AZUMAMIDE B)copy SMILEScopy InChI
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of human HDAC1 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483229(CHEMBL1642815)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetHistone deacetylase 4(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50372469(AZUMAMIDE E)copy SMILEScopy InChI
Affinity DataIC50: 2.28E+3nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483244(CHEMBL1642816)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483241(CHEMBL1642803)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetHistone deacetylase 4(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50377384(AZUMAMIDE C)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetHistone deacetylase 4(Human)
Waseda University

Curated by ChEMBL
LigandPNGBDBM50377383(AZUMAMIDE B)copy SMILEScopy InChI
Affinity DataIC50: 3.66E+3nMAssay Description:Inhibition of human HDAC4 expressed in 293T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3M1GPubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483218(CHEMBL1642770)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483217(CHEMBL1642769)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483219(CHEMBL1642773)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483245(CHEMBL1642789)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483230(CHEMBL1642771)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483242(CHEMBL1642808)copy SMILEScopy InChI
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483234(CHEMBL1642767)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483208(CHEMBL1642804)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482163(CHEMBL1086443)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483235(CHEMBL1642772)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483228(CHEMBL1642787)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483223(CHEMBL1642777)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483199(CHEMBL1642790)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483224(CHEMBL1642781)copy SMILEScopy InChI
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483232(CHEMBL1642788)copy SMILEScopy InChI
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483226(CHEMBL1642784)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483216(CHEMBL1642768)copy SMILEScopy InChI
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50109350(CHEMBL3600948)copy SMILEScopy InChI
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of Influenza A/Perto Rico/8/34 (PR8) (H1N1) PA N-terminal domain (1 to 197) endonuclease activity expressed in Escherichia coli Rosetta (D...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483225(CHEMBL1642783)copy SMILEScopy InChI
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483227(CHEMBL1642785)copy SMILEScopy InChI
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483248(CHEMBL1642779)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483239(CHEMBL1642786)copy SMILEScopy InChI
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483250(CHEMBL1642807)copy SMILEScopy InChI
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetPolymerase acidic protein(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Chiba University

Curated by ChEMBL
LigandPNGBDBM50109353(CHEMBL3600947)copy SMILEScopy InChI
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of Influenza A/Perto Rico/8/34 (PR8) (H1N1) PA N-terminal domain (1 to 197) endonuclease activity expressed in Escherichia coli Rosetta (D...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483237(CHEMBL1642778)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50482163(CHEMBL1086443)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activity after 1 hr by densitometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RT5PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483231(CHEMBL1642780)copy SMILEScopy InChI
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50483215(CHEMBL1642765)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition RNase H activity of HIV1 reverse transcriptase expressed in Escherichia coli stain BL21(DE3)pLysSMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3Q11PubMed
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