Compile Data Set for Download or QSAR
Found 85 with Last Name = 'ikura' and Initial = 't'
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Transrepression of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-NCoR and MH100(UAS) X 4tk-LUC reporter plasmid asse...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M04801PubMedDrugBank
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)copy SMILEScopy InChI
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [3H]-1alpha,25-dihydroxyvitamin D3 from recombinant human VDR LBD expressed in Escherichia coli BL21 (DE3) pLysS after 16 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78H20PubMedDrugBank
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50281390(CHEMBL4159525)copy SMILEScopy InChI
Affinity DataIC50: 0.0900nMAssay Description:Transrepression of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-NCoR and MH100(UAS) X 4tk-LUC reporter plasmid asse...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M04801PubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50135039(CHEMBL3745849)copy SMILEScopy InChI
Affinity DataIC50: 0.0900nMAssay Description:Agonist activity at VDR (unknown origin) expressed in HEK293 cells cotransfected with NCoR assessed as decrease in NCoR recruitment by two-hybrid ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HZCPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Agonist activity at VDR (unknown origin) expressed in HEK293 cells cotransfected with NCoR assessed as decrease in NCoR recruitment by two-hybrid ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HZCPubMedDrugBank
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50129805(CHEMBL3629552)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMAssay Description:Displacement of [3H]-1alpha,25-dihydroxyvitamin D3 from recombinant human VDR LBD expressed in Escherichia coli BL21 (DE3) pLysS after 16 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78H20PubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50281390(CHEMBL4159525)copy SMILEScopy InChI
Affinity DataIC50: 0.240nMAssay Description:Displacement of [26,27-Methyl-3H]-1,25(OH)2D3 from recombinant human GST-tagged VDR LBD (140 to 427 residues) expressed in Escherichia coli BL21 prei...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M04801PubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from recombinant human VDR ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HZCPubMedDrugBank
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50281389(CHEMBL4173602)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Transrepression of VP16-tagged VDR (unknown origin) expressed in HEK293 cells harboring pCMX-GAL4-NCoR and MH100(UAS) X 4tk-LUC reporter plasmid asse...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M04801PubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50292705((25R)-25-Adamantyl-1alpha,25-dihydroxy-2-methylene...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at VDR expressed in COS7 cells assessed as inhibition of 1,25-Dihydroxyvitamin D3-induced response by transient transcription ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9W2ZPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50281389(CHEMBL4173602)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Displacement of [26,27-Methyl-3H]-1,25(OH)2D3 from recombinant human GST-tagged VDR LBD (140 to 427 residues) expressed in Escherichia coli BL21 prei...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M04801PubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50135039(CHEMBL3745849)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from recombinant human VDR ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HZCPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015315(CHEMBL3263870)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015316(CHEMBL3263873)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015317(CHEMBL3263872)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from GST-fused human VDR-LBD expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50135031(CHEMBL3747243)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from recombinant human VDR ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HZCPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50292704((1R,3R,7E,17beta)-17-{(1S,2E,5R)-5-hydroxy-1-methy...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at VDR expressed in COS7 cells assessed as inhibition of 1,25-Dihydroxyvitamin D3-induced response by transient transcription ass...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9W2ZPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50135095(CHEMBL3747761)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from recombinant human VDR ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HZCPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50135094(CHEMBL3745746)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Displacement of [3H]-1,25(OH)2D3 from recombinant human VDR ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2HZCPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50512559(CHEMBL4540985)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Transactivation of VDR in human Macrophage-like cell assessed as cell differentiation measured after 4 days by NBT dye-based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380PQPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244240((20S)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)copy SMILEScopy InChI
Affinity DataEC50:  0.0260nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50412385(CHEMBL2021488)copy SMILEScopy InChI
Affinity DataEC50:  0.0900nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50005618(CHEMBL2021484)copy SMILEScopy InChI
Affinity DataEC50:  0.00210nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244241((20R)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244165((1R,2S,3R,5Z,7E)-17-{(1R)-1-[(2-ethyl-2-hydroxybut...)copy SMILEScopy InChI
Affinity DataEC50:  0.0240nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244269((20R)-1-alpha-2-alpha-25-Trihydroxy-2-beta-methyl-...)copy SMILEScopy InChI
Affinity DataEC50:  0.120nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50412386(CHEMBL2021486)copy SMILEScopy InChI
Affinity DataEC50:  0.0580nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244241((20R)-(2E)-1-alpha-25-Dihydroxy-2-[2-(hydroxy)-eth...)copy SMILEScopy InChI
Affinity DataEC50:  0.0290nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244165((1R,2S,3R,5Z,7E)-17-{(1R)-1-[(2-ethyl-2-hydroxybut...)copy SMILEScopy InChI
Affinity DataEC50:  0.115nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244268((20S)-1-alpha-2-alpha-25-Trihydroxy-2beta-methyl-1...)copy SMILEScopy InChI
Affinity DataEC50:  1.90nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Mus musculus)
Tokyo Medical and Dental University

Curated by ChEMBL
LigandPNGBDBM50244269((20R)-1-alpha-2-alpha-25-Trihydroxy-2-beta-methyl-...)copy SMILEScopy InChI
Affinity DataEC50:  4.5nMAssay Description:Increase in mouse VDR-mediated transcriptional activity in african green monkey COS7 cells after 24 hrs by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60NWWPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015315(CHEMBL3263870)copy SMILEScopy InChI
Affinity DataEC50:  6.60nMAssay Description:Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015316(CHEMBL3263873)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015317(CHEMBL3263872)copy SMILEScopy InChI
Affinity DataEC50:  1.5nMAssay Description:Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)copy SMILEScopy InChI
Affinity DataEC50:  0.0700nMAssay Description:Transactivation of human VDR expressed in HEK293 cells cotransfected with mouse VDRE, Tk-Sppx3-LUC reporter plasmid measured after 24 hrs by lucifera...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015315(CHEMBL3263870)copy SMILEScopy InChI
Affinity DataEC50:  4.40nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)copy SMILEScopy InChI
Affinity DataEC50:  0.600nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015317(CHEMBL3263872)copy SMILEScopy InChI
Affinity DataEC50:  2.30nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015316(CHEMBL3263873)copy SMILEScopy InChI
Affinity DataEC50:  0.800nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-RXRalpha and 4-tk-LUC assessed as heterodimerization with RXRalpha by mammal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015315(CHEMBL3263870)copy SMILEScopy InChI
Affinity DataEC50:  15nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)copy SMILEScopy InChI
Affinity DataEC50:  1.5nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015317(CHEMBL3263872)copy SMILEScopy InChI
Affinity DataEC50:  6.5nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015316(CHEMBL3263873)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-SRC1 and 4-tk-LUC assessed as SRC1 interaction with AF2 surface of VDR by ma...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015315(CHEMBL3263870)copy SMILEScopy InChI
Affinity DataEC50:  4nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)copy SMILEScopy InChI
Affinity DataEC50:  0.400nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015317(CHEMBL3263872)copy SMILEScopy InChI
Affinity DataEC50:  3.70nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015316(CHEMBL3263873)copy SMILEScopy InChI
Affinity DataEC50:  1.80nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-N-CoR and 4-tk-LUC assessed as inhibition of N-CoR binding to VDR by mammali...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015315(CHEMBL3263870)copy SMILEScopy InChI
Affinity DataEC50:  4.10nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-NCoR2 and 4-tk-LUC assessed as inhibition of NCoR2 binding to VDR by mammali...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Universidad de Santiago de Compostela

Curated by ChEMBL
LigandPNGBDBM50015318(CHEMBL3263871)copy SMILEScopy InChI
Affinity DataEC50:  0.5nMAssay Description:Activation of human VDR expressed in HEK293 cells cotransfected CMX-GAL4-NCoR2 and 4-tk-LUC assessed as inhibition of NCoR2 binding to VDR by mammali...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2Z2GPubMed
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