TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 2 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 3.62nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 3 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 3.72nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 2 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 4.11nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 3 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 22.5nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 2 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 23.4nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 2 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 41.7nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 3 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 47.7nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 2 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 53.5nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 3 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKi: 65.9nMAssay Description:Tested for binding affinity against Metabotropic glutamate receptor 3 in CHO cells using [3H]-7 as radioligandMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
TargetCorticotropin-releasing factor receptor 2(RAT)
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Taisho Pharmaceutical Co., Ltd.
Curated by PDSP Ki Database
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Taisho Pharmaceutical Company Ltd.
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:In vitro binding affinity at Sigma opioid receptors on guinea pig brain membranes by [3H]3-PPP displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Escherichia coli TEM1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of Enterobacter cloacae AmpCMore data for this Ligand-Target Pair