Compile Data Set for Download or QSAR
Found 17 with Last Name = 'marumo' and Initial = 't'
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human mGlu3 receptor expressed in CHO cell membranes in presence of glutamate by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human mGlu6 receptor expressed in HEK293T cell membranes in presence of glutamate by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human mGlu4 receptor expressed in CHO cell membranes in presence of glutamate by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human mGlu1 receptor expressed in CHO cell membranes in presence of glutamate by intracellular Ca2+ assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human mGlu8 receptor expressed in CHO cell membranes in presence of glutamate by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at human mGlu2 receptor expressed in CHO cell membranes in presence of glutamate by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50555839(CHEMBL4793451)copy SMILES
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mGlu3 receptor expressed in CHO cell membranes by GTPgammaS binding assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mGlu6 receptor expressed in HEK293T cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mGlu8 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mGlu4 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mGlu1 receptor expressed in CHO cell membranes by intracellular Ca2+ assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50:  153nMAssay Description:Agonist activity at human mGlu2 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 2(Rattus norvegicus)TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50:  154nMAssay Description:Agonist activity at rat mGlu2 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50555839(CHEMBL4793451)copy SMILES
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mGlu3 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50:  76nMAssay Description:Agonist activity at human mGlu3 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50555839(CHEMBL4793451)copy SMILES
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at human mGlu2 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50094841((+)-2-Amino-3-fluoro-bicyclo[3.1.0]hexane-2,6-dica...)copy SMILEScopy InChI
Affinity DataEC50:  97nMAssay Description:Agonist activity at rat mGlu3 receptor expressed in CHO cell membranes by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5Z03PubMed