Compile Data Set for Download or QSAR
Found 187 with Last Name = 'nakahata' and Initial = 't'
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268236(CHEMBL4101718)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492580(CHEMBL2407328)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Mus musculus)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50545129(CHEMBL4645607)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of mouse recombinant C-terminal FLAG-tagged SMS2 expressed in mammalian expression system using C14-phosphatidylcholineD72 and C17-ceramid...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J106QTPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268214(CHEMBL4070852)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Mus musculus)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50545128(CHEMBL4641888)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of mouse recombinant C-terminal FLAG-tagged SMS2 expressed in mammalian expression system using C14-phosphatidylcholineD72 and C17-ceramid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J106QTPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268237(CHEMBL4060964)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268236(CHEMBL4101718)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268214(CHEMBL4070852)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268213(CHEMBL4092798)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268235(CHEMBL4074342)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492572(CHEMBL2407322)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268215(CHEMBL4100114)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492567(CHEMBL2407333)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268216(CHEMBL4060897)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268217(CHEMBL4064789)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268212(CHEMBL4077605)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50282224(CHEMBL4172856)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Compound was evaluated for the inhibition of dihydrofolate reductase obtained from humanMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29G5QB9PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268193(CHEMBL4059929)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268194(CHEMBL4100523)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268217(CHEMBL4064789)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268237(CHEMBL4060964)copy SMILEScopy InChI
Affinity DataIC50: 7.60nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Mus musculus)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50545122(CHEMBL4646354)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Inhibition of mouse recombinant C-terminal FLAG-tagged SMS2 expressed in mammalian expression system using C14-phosphatidylcholineD72 and C17-ceramid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J106QTPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268215(CHEMBL4100114)copy SMILEScopy InChI
Affinity DataIC50: 7.80nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492578(CHEMBL2407320)copy SMILEScopy InChI
Affinity DataIC50: 8.70nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492583(CHEMBL2407319)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492578(CHEMBL2407320)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492584(CHEMBL2407323)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492583(CHEMBL2407319)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268222(CHEMBL4063587)copy SMILEScopy InChI
Affinity DataIC50: 9.60nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492582(CHEMBL2407336)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492584(CHEMBL2407323)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492581(CHEMBL2407334)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492582(CHEMBL2407336)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268219(CHEMBL4073378)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268220(CHEMBL4094029)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Mus musculus)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50545127(CHEMBL4644293)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of mouse recombinant C-terminal FLAG-tagged SMS2 expressed in mammalian expression system using C14-phosphatidylcholineD72 and C17-ceramid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J106QTPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492573(CHEMBL2407332)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268220(CHEMBL4094029)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited

Curated by ChEMBL
LigandPNGBDBM50282208(CHEMBL4177314)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Compound was evaluated for the inhibition of Folyl-polyglutamate synthase obtained from porcineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29G5QB9PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492575(CHEMBL2407337)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492585(CHEMBL2407326)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268218(CHEMBL4086265)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492572(CHEMBL2407322)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetPhosphatidylcholine:ceramide cholinephosphotransferase 2(Mus musculus)
Takeda Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50545123(CHEMBL4638337)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of mouse recombinant C-terminal FLAG-tagged SMS2 expressed in mammalian expression system using C14-phosphatidylcholineD72 and C17-ceramid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J106QTPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268219(CHEMBL4073378)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492567(CHEMBL2407333)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492574(CHEMBL2407325)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Displacement of [3H]-hydroxytryptamine from human SERT expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Takeda Pharmaceutical Company Ltd

Curated by ChEMBL
LigandPNGBDBM50492579(CHEMBL2407327)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]-norepinephrine from human NET expressed in CHO cells by TopCounting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2DVQPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268216(CHEMBL4060897)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
TargetSomatostatin receptor type 5(Mus musculus)
Research Division, Takeda Pharmaceutical Co., Ltd., 26-1, Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. Electronic address: takeshi.yamasaki@takeda.com.

Curated by ChEMBL
LigandPNGBDBM50268212(CHEMBL4077605)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Antagonist activity at mouse SSTR5 expressed in CHO cells assessed as inhibition of SST14-induced forskolin-stimulated intracellular cAMP level incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8P5GPubMed
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