Compile Data Set for Download or QSAR
Found 94 with Last Name = 'nishioka' and Initial = 't'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50509099(CHEMBL4565294)copy SMILEScopy InChI
Affinity DataKi:  7.27E+4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WZTPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50509099(CHEMBL4565294)copy SMILEScopy InChI
Affinity DataKi:  2.20E+5nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WZTPubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50509099(CHEMBL4565294)copy SMILEScopy InChI
Affinity DataKi:  1.43E+6nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WZTPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50509101(CHEMBL4460098)copy SMILEScopy InChI
Affinity DataKi:  2.47E+6nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WZTPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50509101(CHEMBL4460098)copy SMILEScopy InChI
Affinity DataKi:  3.73E+6nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WZTPubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Eisai Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50509101(CHEMBL4460098)copy SMILEScopy InChI
Affinity DataKi:  1.21E+7nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in rat brain after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WZTPubMed
LigandPNGBDBM50116000((S)-3-{(12R,13R)-13-Hydroxy-13-[(4R,2'R,5'R)-5'-((...)copy SMILEScopy InChI
Affinity DataIC50: 0.75nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC8290PubMed
LigandPNGBDBM50366820(BULLATACIN)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58MWCPubMed
LigandPNGBDBM50116000((S)-3-{(12R,13R)-13-Hydroxy-13-[(4R,2'R,5'R)-5'-((...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58MWCPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92960(Piperazine derivative, 24)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
LigandPNGBDBM50130144(2-{(12R,13R)-13-Hydroxy-13-[(4R,2'R,5'R)-5'-((R)-1...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58MWCPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92945(Piperazine derivative, 10)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92946(Piperazine derivative, 9)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411085(CHEMBL464549)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92949(Piperazine derivative, 13)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92955(Piperazine derivative, 19)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92948(Piperazine derivative, 12)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92941(Piperazine derivative, 5)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
LigandPNGBDBM50139593((S)-3-{13-[(2R,5S,1'R,3'R)-5'-((R)-1-Hydroxy-undec...)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC8290PubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92950(Piperazine derivative, 14)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
LigandPNGBDBM50139595((S)-3-[(R)-13-Hydroxy-13-((2R,5R,1'S,3'R)-5'-undec...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC8290PubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411084(CHEMBL208839)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92956(Piperazine derivative, 20)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92947(Piperazine derivative, 11)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411092(CHEMBL209302)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411088(CHEMBL211108)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92944(Piperazine derivative, 8)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92954(Piperazine derivative, 18)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92942(Piperazine derivative, 6)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411091(CHEMBL377863)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411087(CHEMBL377013)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411082(CHEMBL208980)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411083(CHEMBL379529)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
LigandPNGBDBM50139594((S)-5-Methyl-3-[13-((2R,5S,1'S,3'R)-5'-undecyl-oct...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibitory concentration needed to halve the control NADH oxidase activity in bovine heart submitochondrial particles (SMP)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZC8290PubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92943(Piperazine derivative, 7)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411093(CHEMBL211884)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
LigandPNGBDBM50130145((R)-1-[(5R,2'R,5'R)-5'-((R)-1-Hydroxy-undecyl)-oct...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58MWCPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411089(CHEMBL211178)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92951(Piperazine derivative, 15)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411090(CHEMBL211345)copy SMILEScopy InChI
Affinity DataIC50: 870nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92953(Piperazine derivative, 17)copy SMILEScopy InChI
Affinity DataIC50: 930nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92958(Piperazine derivative, 22)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92957(Piperazine derivative, 21)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50411086(CHEMBL378692)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
LigandPNGBDBM50130143((R)-1-[(2R,5R,2'R,5'R)-5'-((R)-1-hydroxy-hexyl)-oc...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of complex I activity was determined by NADH oxidase assay using bovine heart submitochondrial particles.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2N58MWCPubMed
TargetAcyl carrier protein, mitochondrial(Bos taurus)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50130143((R)-1-[(2R,5R,2'R,5'R)-5'-((R)-1-hydroxy-hexyl)-oc...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of bovine mitochondrial NADH-ubiquinone oxidoreductase by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60Q8NPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92959(Piperazine derivative, 23)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92940(Piperazine derivative, 4)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))
Kyoto University

LigandPNGBDBM92952(Piperazine derivative, 16)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition assay using NADH-ubiquinone oxidoreductase (complex I).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50KKQPubMed
TargetSucrase-isomaltase, intestinal(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50009001(5,6,7-Trihydroxyflavone | 5,6,7-trihydroxy-2-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human intestinal sucrase in human Caco2 cell membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1CFBPubMed
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