Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GSK-3-beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GSK-3-beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p38alpha MAPK expressed in baculovirus infected Sf9 insect cells using p38 peptide ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibition of NanoBRET kinase tracer K4 binding to full-length human C-terminal NanoLuc-tagged p38alpha MAPK expressed in HEK293T cells incubated for...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of NanoBRET kinase tracer K4 binding to full-length human C-terminal NanoLuc-tagged p38alpha MAPK expressed in HEK293T cells incubated for...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human GSK-3-beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant human GSK-3-beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of NanoBRET kinase tracer K4 binding to full-length human C-terminal NanoLuc-tagged p38alpha MAPK expressed in HEK293T cells incubated for...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
In DepthDetails
Affinity DataIC50: 11nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p38alpha MAPK expressed in baculovirus infected Sf9 insect cells using p38 peptide ...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p38alpha MAPK expressed in baculovirus infected Sf9 insect cells using p38 peptide ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of NanoBRET kinase tracer K4 binding to full-length human C-terminal NanoLuc-tagged p38alpha MAPK expressed in HEK293T cells incubated for...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Competitive inhibition of human recombinant full length GSK3beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated with enzyme for 10 min...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p38alpha MAPK expressed in baculovirus infected Sf9 insect cells using p38 peptide ...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of GSK3beta (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant human GSK-3-beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of P38alpha MAPK (unknown origin) by ADP-Glo assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged p38alpha MAPK expressed in baculovirus infected Sf9 insect cells using p38 peptide ...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant human GSK-3-beta using YRRAAVPPSPSLSRHSSPHQ(pS)EDEEE as substrate preincubated for 10 mins followed by substrate addition a...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Eberhard Karls Universit£t T£bingen
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
Ligand Info
In DepthDetails
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