Compile Data Set for Download or QSAR
Found 254 with Last Name = 'rossi' and Initial = 't'
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50408664(GR-205171 | VOFOPITANT)copy SMILEScopy InChI
Affinity DataKi:  0.0501nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50020217((4aR,10bR)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-na...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Agonistic activity at DRD3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413891(VESTIPITANT)copy SMILEScopy InChI
Affinity DataKi:  0.224nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413892(CHEMBL490926)copy SMILEScopy InChI
Affinity DataKi:  0.427nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413890(CHEMBL492117 | TCMDC-138495)copy SMILEScopy InChI
Affinity DataKi:  0.537nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414563(CHEMBL559873)copy SMILEScopy InChI
Affinity DataKi:  0.631nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Antagonistic activity at human DRD3 receptor by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50331549(CHEMBL567286 | [11C]-3-(2-oxo-3-(2-(4-(trifluorome...)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Antagonistic activity at rat DRD3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414574(CHEMBL563580)copy SMILEScopy InChI
Affinity DataKi:  1.26nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413892(CHEMBL490926)copy SMILEScopy InChI
Affinity DataKi:  1.29nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414578(CHEMBL558058)copy SMILEScopy InChI
Affinity DataKi:  1.58nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50411402(CHEMBL244946)copy SMILEScopy InChI
Affinity DataKi:  1.58nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414570(CHEMBL563635)copy SMILEScopy InChI
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414403(CHEMBL560177)copy SMILEScopy InChI
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414557(CHEMBL562464)copy SMILEScopy InChI
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414572(CHEMBL563860)copy SMILEScopy InChI
Affinity DataKi:  2.51nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414555(CHEMBL565075)copy SMILEScopy InChI
Affinity DataKi:  3.16nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414563(CHEMBL559873)copy SMILEScopy InChI
Affinity DataKi:  3.16nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413888(CHEMBL523156)copy SMILEScopy InChI
Affinity DataKi:  3.72nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50370572(CHEMBL85606 | SB-277011)copy SMILEScopy InChI
Affinity DataKi:  3.98nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414572(CHEMBL563860)copy SMILEScopy InChI
Affinity DataKi:  3.98nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414574(CHEMBL563580)copy SMILEScopy InChI
Affinity DataKi:  5.01nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414566(CHEMBL563435)copy SMILEScopy InChI
Affinity DataKi:  5.01nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414565(CHEMBL563274)copy SMILEScopy InChI
Affinity DataKi:  6.31nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50020217((4aR,10bR)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-na...)copy SMILEScopy InChI
Affinity DataKi:  6.31nMAssay Description:Agonistic activity at DRD2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413889(CHEMBL489924)copy SMILEScopy InChI
Affinity DataKi:  8.13nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413894(CHEMBL521605)copy SMILEScopy InChI
Affinity DataKi:  8.71nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414567(CHEMBL562948)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414571(CHEMBL563563)copy SMILEScopy InChI
Affinity DataKi:  12.6nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414554(CHEMBL551927)copy SMILEScopy InChI
Affinity DataKi:  15.8nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414556(CHEMBL564930)copy SMILEScopy InChI
Affinity DataKi:  15.8nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetSubstance-P receptor(Homo sapiens (Human))
GlaxoSmithKline Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50413893(CHEMBL522292)copy SMILEScopy InChI
Affinity DataKi:  18.2nMAssay Description:Displacement of [3H]substance P from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0425PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414554(CHEMBL551927)copy SMILEScopy InChI
Affinity DataKi:  19.9nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414578(CHEMBL558058)copy SMILEScopy InChI
Affinity DataKi:  19.9nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414581(CHEMBL560270)copy SMILEScopy InChI
Affinity DataKi:  19.9nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414579(CHEMBL564948)copy SMILEScopy InChI
Affinity DataKi:  25.1nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414564(CHEMBL562833)copy SMILEScopy InChI
Affinity DataKi:  25.1nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414555(CHEMBL565075)copy SMILEScopy InChI
Affinity DataKi:  25.1nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414558(CHEMBL556496)copy SMILEScopy InChI
Affinity DataKi:  25.1nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414557(CHEMBL562464)copy SMILEScopy InChI
Affinity DataKi:  25.1nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414570(CHEMBL563635)copy SMILEScopy InChI
Affinity DataKi:  25.1nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetThymidylate synthase(Homo sapiens (Human))
UNIMORE

LigandPNGBDBM18771((2S)-2-[(4-{[(2-amino-4-oxo-1,4-dihydroquinazolin-...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:TS was assayed spectrophotometrically in the reaction buffer solution containing (6R, 6S)-5, 10-CH2H4folate. The reaction was initiated by the additi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S180R0PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414562(CHEMBL554738)copy SMILEScopy InChI
Affinity DataKi:  31.6nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414556(CHEMBL564930)copy SMILEScopy InChI
Affinity DataKi:  31.6nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414568(CHEMBL562836)copy SMILEScopy InChI
Affinity DataKi:  39.8nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414987(CHEMBL567919)copy SMILEScopy InChI
Affinity DataKi:  50.1nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414560(CHEMBL563926)copy SMILEScopy InChI
Affinity DataKi:  50.1nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414575(CHEMBL561128)copy SMILEScopy InChI
Affinity DataKi:  50.1nMAssay Description:Binding affinity to human DRD3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Imperial College London

Curated by ChEMBL
LigandPNGBDBM50414562(CHEMBL554738)copy SMILEScopy InChI
Affinity DataKi:  50.1nMAssay Description:Binding affinity to human DRD2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7X7CPubMed
TargetThymidylate synthase(Lactobacillus casei)
UNIMORE

LigandPNGBDBM18771((2S)-2-[(4-{[(2-amino-4-oxo-1,4-dihydroquinazolin-...)copy SMILEScopy InChI
Affinity DataKi:  60nM ΔG°:  -40.5kJ/molepH: 7.4 T: 2°CAssay Description:TS was assayed spectrophotometrically in the reaction buffer solution containing (6R, 6S)-5, 10-CH2H4folate. The reaction was initiated by the additi...More data for this Ligand-Target Pair
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