TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Novartis Takarazuka Research Institute
Curated by ChEMBL
Novartis Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 134nMAssay Description:TP_TRANSPORTER: inhibition of ATPase activity (Verapamil) in P-gp-MRP-16-Protein A complexMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Novartis Takarazuka Research Institute
Curated by ChEMBL
Novartis Takarazuka Research Institute
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:TP_TRANSPORTER: inhibition of Taxol transepithelial transport (basal to apical) in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of Vitronectin binding to GPIIb/IIIIa Vitronectin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of vWF binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of vWF binding to GPIIb/IIIIa receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Vitronectin binding to GPIIb/IIIIa Vitronectin receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:TP_TRANSPORTER: drug resistance(Mitoxantrone) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:TP_TRANSPORTER: drug resistance(SN-38) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Inhibition of biotinylated fibrinogen binding to alphaIIb-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:TP_TRANSPORTER: drug resistance(Mitoxantrone) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:TP_TRANSPORTER: drug resistance(SN-38) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:TP_TRANSPORTER: drug resistance(SN-38) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:TP_TRANSPORTER: drug resistance(Mitoxantrone) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:TP_TRANSPORTER: drug resistance(Mitoxantrone) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:TP_TRANSPORTER: drug resistance(Mitoxantrone) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:TP_TRANSPORTER: drug resistance(SN-38) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Japanese Foundation for Cancer Research
Curated by ChEMBL
Japanese Foundation for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:TP_TRANSPORTER: drug resistance(SN-38) in BCRP-expressing K562 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Biotinylated fibrinogen binding to alpha IIb beta3 integrinMore data for this Ligand-Target Pair
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