Compile Data Set for Download or QSAR
Found 389 with Last Name = 'nguyen' and Initial = 'tb'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)

Curated by ChEMBL
LigandPNGBDBM50383311(CHEMBL2029619)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GHWPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)

Curated by ChEMBL
LigandPNGBDBM50383305(CHEMBL2029615)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GHWPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GHWPubMedDrugBank
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)

Curated by ChEMBL
LigandPNGBDBM50383306(CHEMBL2029618)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GHWPubMed
TargetTranscription factor p65(Homo sapiens (Human))
MediQuest Therapeutics, Inc.

Curated by ChEMBL
LigandPNGBDBM50195806(CHEMBL384590 | N-(3-(4-(3-aminopropylamino)butylam...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of NFkappaB in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34X4HPubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)

Curated by ChEMBL
LigandPNGBDBM50383304(CHEMBL2029622)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GHWPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut de Chimie des Substances Naturelles (ICSN)

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0GHWPubMed
TargetTranscription factor p65(Homo sapiens (Human))
MediQuest Therapeutics, Inc.

Curated by ChEMBL
LigandPNGBDBM50195808(CHEMBL218163 | N-(3-(4-(3-aminopropylamino)butylam...)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of NFkappaB in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34X4HPubMed
TargetTranscription factor p65(Homo sapiens (Human))
MediQuest Therapeutics, Inc.

Curated by ChEMBL
LigandPNGBDBM50195809(CHEMBL218434 | N-(3-(4-(3-aminopropylamino)butylam...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of NFkappaB in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34X4HPubMed
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366340(US9873693, Compound 268)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366341(US9873693, Compound 269)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366187(US9873693, Compound 110 | US9873693, Compound 270 ...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366343(US9873693, Compound 271)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366344(US9873693, Compound 272)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366345(US9873693, Compound 273)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366240(US9873693, Compound 163)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366241(US9873693, Compound 164)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366242(US9873693, Compound 165)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366243(US9873693, Compound 166)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366245(US9873693, Compound 168)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366246(US9873693, Compound 169)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366190(US9873693, Compound 113 | US9873693, Compound 274)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366156(US9873693, Compound 79)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366157(US9873693, Compound 80)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366158(US9873693, Compound 81)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366159(US9873693, Compound 82)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366160(US9873693, Compound 83)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366161(US9873693, Compound 84)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366162(US9873693, Compound 85)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366247(US9873693, Compound 170)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366248(US9873693, Compound 171)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366196(US9873693, Compound 119 | US9873693, Compound 276)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366202(US9873693, Compound 125 | US9873693, Compound 277)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366163(US9873693, Compound 86)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366164(US9873693, Compound 87)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366165(US9873693, Compound 88)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366166(US9873693, Compound 89)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366167(US9873693, Compound 90)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366168(US9873693, Compound 91)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366169(US9873693, Compound 92)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366350(US9873693, Compound 278)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366351(US9873693, Compound 279)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366352(US9873693, Compound 280)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366170(US9873693, Compound 93)copy SMILES
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366171(US9873693, Compound 94)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366172(US9873693, Compound 95)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366173(US9873693, Compound 96)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366174(US9873693, Compound 97)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366175(US9873693, Compound 98)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM366249(US9873693, Compound 172)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H41TRTUS Patent
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