TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of NFkappaB in human HEK293 cellsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of human recombinant CDK5/p25 using [gamma 33P]ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Institut de Chimie des Substances Naturelles (ICSN)
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of GST-tagged rat recombinant DYRK1A expressed in Escherichia coli using KKISGRLSPIMTEQ as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of NFkappaB in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of NFkappaB in human HEK293 cellsMore data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1 [51-360](Homo sapiens (Human))
Duquesne University
Duquesne University
Affinity DataIC50: 500nMAssay Description:A PDK1 kinase assay was performed as follows. PDK1 (amino acids 51-360) and AKT2 (amino acids 140-467 fused to PIFtide, amino acids EEQEMFRDFDYIADW) ...More data for this Ligand-Target Pair
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