Compile Data Set for Download or QSAR
Found 186 with Last Name = 'somervaille' and Initial = 'tcp'
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241539(CHEMBL4084845)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Kinetic constant was measured for PMII of Leishmania donovani promastigotes using supernatant (S12) fractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262048(CHEMBL3134377)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242934(CHEMBL4066743)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of platelet aggregation (PRP)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262023(CHEMBL4071991)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242954(CHEMBL4101067)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241533(CHEMBL4102775)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242894(CHEMBL4074323)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM301063(4-{3-[((3R)-3- aminopiperidyl)carbonyl]-5-(2- pyri...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of full length human LSD1 expressed in Escherichia coli using H3K4me1-biotin labeled peptide as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242895(CHEMBL4076163)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of platelet aggregation (PRP)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242950(CHEMBL4074334)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242905(CHEMBL4103503)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of Fibrinogen receptor bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242892(CHEMBL4088045)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262052(CHEMBL4066130)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241526(CHEMBL4095018)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242886(CHEMBL4104407)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM301063(4-{3-[((3R)-3- aminopiperidyl)carbonyl]-5-(2- pyri...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262070(CHEMBL4092760)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242952(CHEMBL4088035)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241535(CHEMBL4068129)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibitory activity against human immunodeficiency virus-1 reverse transcriptase(HIV-1 RT).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242953(CHEMBL4066749)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241531(CHEMBL4095517)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Binding potency against Vasopressin V1 receptor in rat liver cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242907(CHEMBL4077730)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242905(CHEMBL4103503)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of LSD1 in human THP1 cells assessed as upregulation of CD86 levels by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241520(CHEMBL4064882)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242934(CHEMBL4066743)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of Fibrinogen receptor bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242883(CHEMBL4062785)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242954(CHEMBL4101067)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Inhibition of LSD1 in human THP1 cells assessed as upregulation of CD86 levels by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262045(CHEMBL4087724)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241493(CHEMBL4103264)copy SMILEScopy InChI
Affinity DataIC50: 620nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242891(CHEMBL4095768)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242890(CHEMBL4077739)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262071(CHEMBL4100487)copy SMILEScopy InChI
Affinity DataIC50: 680nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242948(CHEMBL4082935)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242889(CHEMBL4069461)copy SMILEScopy InChI
Affinity DataIC50: 720nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242956(CHEMBL4085581)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of Fibrinogen receptor bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241495(CHEMBL4079933)copy SMILEScopy InChI
Affinity DataIC50: 810nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262044(CHEMBL4082476)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241534(CHEMBL4074550)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262074(CHEMBL4105603)copy SMILEScopy InChI
Affinity DataIC50: 950nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241523(CHEMBL4084823)copy SMILEScopy InChI
Affinity DataIC50: 990nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241527(CHEMBL4098894)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242951(CHEMBL4096682)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50262072(CHEMBL4079770)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using histone H3(1-21)K4(Me1) biotin pe...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28918CTPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242896(CHEMBL4093330)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242887(CHEMBL4080173)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241497(CHEMBL4087810)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241528(CHEMBL4071901)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242885(CHEMBL4101077)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242945(CHEMBL4073624)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241519(CHEMBL4073481)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of N-terminal truncated human LSD1 (151 to 852 residues) expressed in Escherichia coli after 30 mins using histone H3(1-21)K4(Me1) biotin ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M32XX8PubMed
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