Compile Data Set for Download or QSAR
Found 15 with Last Name = 'coetzer' and Initial = 'tl'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in peak channel current by IonWork patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1H22PubMedDrugBank
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50030836(CHEMBL3355639)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SJDPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50129589(CHEMBL3628223)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SJDPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50129559(CHEMBL3234071)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SJDPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50129562(CHEMBL3628220)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SJDPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50563339(CHEMBL4756352)copy SMILES
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N84VCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50563340(CHEMBL4743418)copy SMILES
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N84VCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50129560(CHEMBL3628216)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SJDPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50518587(CHEMBL4459380)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in peak channel current by IonWork patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1H22PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50518589(CHEMBL4468890)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in peak channel current by IonWork patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1H22PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50518586(CHEMBL4457843)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in peak channel current by IonWork patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1H22PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50518585(CHEMBL4466654)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in peak channel current by IonWork patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1H22PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50518588(CHEMBL4576616)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells assessed as reduction in peak channel current by IonWork patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1H22PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50563338(CHEMBL4764956)copy SMILES
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERG incubated for 4 hrs by fluorescene microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N84VCPubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Cape Town

Curated by ChEMBL
LigandPNGBDBM50129561(CHEMBL3628219)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ERG potassium channel by ionworks patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SJDPubMed