Compile Data Set for Download or QSAR
Found 74 with Last Name = 'bocan' and Initial = 'tm'
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50011204(CHEMBL2368094 | Sodium; 7-[4-(4-fluoro-phenyl)-2-i...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50006407(CHEMBL2367472 | Sodium; 7-[5-(4-fluoro-phenyl)-3-i...)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50006409(CHEMBL2367478 | Sodium; 7-[5-(4-fluoro-phenyl)-3-i...)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50011213(CHEMBL3349878 | Sodium; 7-[2-(4-fluoro-phenyl)-5-i...)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50011211(CHEMBL2368089 | Sodium; 7-[4-(4-fluoro-phenyl)-2-i...)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063243(CHEMBL161499 | N-(2,6-Diisopropyl-phenyl)-2-pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50011208(7-[4-(4-Fluoro-phenyl)-2-isopropyl-6-methyl-1-oxy-...)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
TargetLiver carboxylesterase 1(Oryctolagus cuniculus (rabbit))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063239(CHEMBL161638 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase by microsomal LAI assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50006410(CHEMBL2367477 | Sodium; 7-[5-(4-fluoro-phenyl)-3-i...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063239(CHEMBL161638 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063226(CHEMBL160149 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063236(CHEMBL159871 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063231(CHEMBL159621 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50014345(CHEMBL11804 | Sodium; (E)-(3R,5S)-9,9-bis-(4-fluor...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50011206(2-Methyl-butyric acid 8-[2-(4-hydroxy-6-oxo-tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063235(CHEMBL161798 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063232(2-Phenyl-N-(2,4,6-trimethoxy-phenyl)-malonamic aci...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063229(CHEMBL161292 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063220(CHEMBL161270 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053404(CHEMBL340148 | N-(2,6-Diisopropyl-phenyl)-2-(5-dod...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053395(2-(3-Dodecyl-isoxazol-5-yl)-2-phenyl-N-(2,4,6-trim...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287512(3-(2,6-Diisopropyl-phenyl)-1-phenyl-1-{2-[8-(tetra...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Liver Acyl coenzyme A:cholesterol acyltransferase inhibitory activity was determined in vitro using [1-14C]-oleolyl-CoA and microsomes isolated from ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZF6
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063221(CHEMBL161295 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053394(2-(5-Dodecyl-[1,3,4]oxadiazol-2-yl)-2-phenyl-N-(2,...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053399(CHEMBL339119 | N-(2,6-Diisopropyl-phenyl)-2-(3-dod...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetLiver carboxylesterase 1(Oryctolagus cuniculus (rabbit))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063239(CHEMBL161638 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase by microsomal MAI2 assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063227(2-Phenyl-N-(2,4,6-trimethoxy-phenyl)-malonamic aci...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063230(CHEMBL159491 | N-(2,6-Diisopropyl-phenyl)-2,2-dime...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053406(2-(4-Dodecyl-[1,2,3]triazol-1-yl)-2-phenyl-N-(2,4,...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053398(2-(5-Dodecyl-isoxazol-3-yl)-2-phenyl-N-(2,4,6-trim...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063224(CHEMBL159414 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053407(CHEMBL338751 | N-(2,6-Diisopropyl-phenyl)-2-(5-dod...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50011203(CHEMBL3349880 | Sodium; 7-[3,4-dibromo-2-(4-fluoro...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063237(2-Phenyl-N-(2,4,6-trimethoxy-phenyl)-malonamic aci...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287511(1-Cyclohexyl-3-(2,6-diisopropyl-phenyl)-1-(2-dodec...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Liver Acyl coenzyme A:cholesterol acyltransferase inhibitory activity was determined in vitro using [1-14C]-oleolyl-CoA and microsomes isolated from ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZF6
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053405(2-(5-Dodecyl-[1,2,4]oxadiazol-3-yl)-2-phenyl-N-(2,...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053400(2-(3-Dodecyl-[1,2,4]oxadiazol-5-yl)-2-phenyl-N-(2,...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063240(CHEMBL161639 | N-(2,6-Diisopropyl-phenyl)-2-fluoro...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053392(2-(3-Dodecyl-isoxazol-5-yl)-N-(2,4,6-trimethoxy-ph...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50368147((+)-(3R,5S)-fluvastatin | (3R,5S)-fluvastatin | (3...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287513(1-Benzyl-1-(2-dodecyl-2H-tetrazol-5-yl)-3-(2,4,6-t...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Liver Acyl coenzyme A:cholesterol acyltransferase inhibitory activity was determined in vitro using [1-14C]-oleolyl-CoA and microsomes isolated from ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZF6
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063233(CHEMBL159597 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287509(1-[2-(10-Methyl-undecyl)-2H-tetrazol-5-yl]-1-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Liver Acyl coenzyme A:cholesterol acyltransferase inhibitory activity was determined in vitro using [1-14C]-oleolyl-CoA and microsomes isolated from ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZF6
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063234(CHEMBL351398 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Rattus norvegicus (rat))
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50368146(CS-514 | Eptastatin Sodium | PRAVASTATIN SODIUM | ...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Ability to inhibit microsomal preparation of HMG-CoA reductase in rat liver.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2MS3TC4PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287515(1-Phenyl-1-{2-[8-(tetrahydro-pyran-2-yloxy)-octyl]...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Liver Acyl coenzyme A:cholesterol acyltransferase inhibitory activity was determined in vitro using [1-14C]-oleolyl-CoA and microsomes isolated from ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZF6
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053393(2-(4-Dodecyl-pyrazol-1-yl)-2-phenyl-N-(2,4,6-trime...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50287517(3-(2,6-Diisopropyl-phenyl)-1-(2-dodecyl-2H-tetrazo...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Liver Acyl coenzyme A:cholesterol acyltransferase inhibitory activity was determined in vitro using [1-14C]-oleolyl-CoA and microsomes isolated from ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZF6
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50063222(CHEMBL159993 | N-(2,6-Diisopropyl-phenyl)-2-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition in hepatic microsomes isolated from cholesterol-fed ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28051R8PubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Warner-Lambert Company

Curated by ChEMBL
LigandPNGBDBM50053403(CHEMBL125407 | N-(2,4-Difluoro-phenyl)-2-(3-dodecy...)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Inhibition of Acyl coenzyme A:cholesterol acyltransferase 1 from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7NMMPubMed
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