TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 7.85nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1 [1068-1325](Homo sapiens (Human))
INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (THE)
US Patent
INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL (THE)
US Patent
Affinity DataIC50: 12nMAssay Description:Tankyrase activity was assayed using a 96-well format HT Universal Chemiluminescent PARP Assay Kit (Trevigen, Inc, cat. no. 4676-096-K) according to ...More data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 13.3nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex Ltd.
Curated by ChEMBL
Domainex Ltd.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Case Western Reserve University
US Patent
Case Western Reserve University
US Patent
Affinity DataIC50: 15nMpH: 7.5Assay Description:Kinase inhibition assays (10 μL) were performed at 20° C. in 384-well plate format. Compound IC50 values were determined at the apparent Km for ...More data for this Ligand-Target Pair
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